Compile Data Set for Download or QSAR
Found 39 with Last Name = 'gatti iou' and Initial = 'm'
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522280(US11161839, Example 10a)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of BCOR peptide binding to human BCL6 expressed in Escherichia coli measured after 270 mins by BCOR ULight TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522280(US11161839, Example 10a)copy SMILES
Affinity DataIC50: 26nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522280(US11161839, Example 10a)copy SMILES
Affinity DataIC50: 26nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50546197(CHEMBL4755229)copy SMILES
Affinity DataIC50: 30nMAssay Description:Inhibition of BCOR peptide binding to human BCL6 expressed in Escherichia coli measured after 270 mins by BCOR ULight TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587565(CHEMBL5081226)copy SMILES
Affinity DataIC50: 46nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522284(US11161839, Example 10e)copy SMILES
Affinity DataIC50: 54nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522285(US11161839, Example 10f)copy SMILES
Affinity DataIC50: 73nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522286(US11161839, Example 10g)copy SMILES
Affinity DataIC50: 82nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522196(US11161839, Example 1a | US11161839, Example 1b)copy SMILES
Affinity DataIC50: 140nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522291(US11161839, Example 10l)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522235(US11161839, Example 3p)copy SMILES
Affinity DataIC50: 250nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522312(US11161839, Example 11i)copy SMILES
Affinity DataIC50: 320nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522274(US11161839, Example 9l)copy SMILES
Affinity DataIC50: 350nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522311(US11161839, Example 11h)copy SMILES
Affinity DataIC50: 420nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587565(CHEMBL5081226)copy SMILES
Affinity DataIC50: 470nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587560(CHEMBL5079024)copy SMILES
Affinity DataIC50: 550nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522280(US11161839, Example 10a)copy SMILES
Affinity DataIC50: 570nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587564(CHEMBL5089812)copy SMILES
Affinity DataIC50: 790nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522227(US11161839, Example 3l)copy SMILES
Affinity DataIC50: 870nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522266(US11161839, Example 9c)copy SMILES
Affinity DataIC50: 880nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522237(US11161839, Example 4)copy SMILES
Affinity DataIC50: 900nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522226(US11161839, Example 1p)copy SMILES
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522285(US11161839, Example 10f)copy SMILES
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587562(CHEMBL5076223)copy SMILES
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522284(US11161839, Example 10e)copy SMILES
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587554(CHEMBL5090262)copy SMILES
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522196(US11161839, Example 1a | US11161839, Example 1b)copy SMILES
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587558(CHEMBL5079963)copy SMILES
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587559(CHEMBL5088786)copy SMILES
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587557(CHEMBL5080619)copy SMILES
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522312(US11161839, Example 11i)copy SMILES
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587556(CHEMBL5080184)copy SMILES
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587555(CHEMBL5090408)copy SMILES
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587561(CHEMBL5075468)copy SMILES
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587552(CHEMBL5084602)copy SMILES
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522311(US11161839, Example 11h)copy SMILES
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587553(CHEMBL5081011)copy SMILES
Affinity DataIC50: 5.57E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R21585PubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM50587563(CHEMBL5080163)copy SMILES
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetB-cell lymphoma 6 protein(Homo sapiens)TBA
LigandPNGBDBM522280(US11161839, Example 10a)copy SMILES
Affinity DataKd:  234nMAssay Description:Binding affinity to human BCL6 BDB domain by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB