Compile Data Set for Download or QSAR
Found 64 with Last Name = 'janeczko' and Initial = 'm'
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34055(iodinated benzimidazole, 21)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  77nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359847(CHEMBL1928909)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  97nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  133nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359847(CHEMBL1928909)copy SMILEScopy InChI
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  143nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  154nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  172nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359845(CHEMBL1928908)copy SMILEScopy InChI
Affinity DataKi:  188nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359845(CHEMBL1928908)copy SMILEScopy InChI
Affinity DataKi:  195nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  212nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34055(iodinated benzimidazole, 21)copy SMILEScopy InChI
Affinity DataKi:  261nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  266nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156669(4,5,6,7-TETRABROMO-BENZIMIDAZOLE | 4,5,6,7-tetrabr...)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156669(4,5,6,7-TETRABROMO-BENZIMIDAZOLE | 4,5,6,7-tetrabr...)copy SMILEScopy InChI
Affinity DataKi:  315nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
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