Compile Data Set for Download or QSAR
Found 32 with Last Name = 'khattab' and Initial = 'm'
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50263771(1-benzoyl-3-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(...)copy SMILEScopy InChI
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)copy SMILEScopy InChI
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)copy SMILEScopy InChI
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)copy SMILEScopy InChI
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)copy SMILEScopy InChI
Affinity DataKi:  2.29E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291874(CHEMBL4159805)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50292371(CHEMBL4171617)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by CoA reductase inhibition screen (COR) in ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50287578(CHEMBL4167715)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291880(CHEMBL4164161)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291882(CHEMBL4160772)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291876(CHEMBL4165274)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat frontal cortex using [3H]8-OH-DPAT as a radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291877(CHEMBL4175894)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Binding affinity against 5-HT1B receptor in rat brain membrane using [3H]8-OH-DPAT as a selective ligand.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291878(CHEMBL4161839)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50163251(2-(4-(4-hydroxyphenylthio)phenyl)-1H-benzo[d]imida...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291881(CHEMBL4168692)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against purified human plasma renin at pH 6.0More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50291879(CHEMBL4172486)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50292365(CHEMBL4160383)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50292370(CHEMBL4170989)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of Chk2 (unknown origin) assessed as decrease in Cdc25C phosphorylation at Ser216 by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ643KPubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50065965(5-Chloro-1H-indole-2-carboxylic acid ((1S,2R)-1-be...)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196903(CHEMBL3916767)copy SMILEScopy InChI
Affinity DataIC50: 178nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using 10 mM of glucose-1-phosphate as substrate preincubated for 60 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196903(CHEMBL3916767)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196901(CHEMBL3986514)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196912(CHEMBL3969601)copy SMILEScopy InChI
Affinity DataIC50: 3.24E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196904(CHEMBL3952333)copy SMILEScopy InChI
Affinity DataIC50: 3.58E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196909(CHEMBL3915666)copy SMILEScopy InChI
Affinity DataIC50: 3.97E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196911(CHEMBL3932944)copy SMILEScopy InChI
Affinity DataIC50: 4.02E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196908(CHEMBL3897672)copy SMILEScopy InChI
Affinity DataIC50: 4.37E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196906(CHEMBL3925760)copy SMILEScopy InChI
Affinity DataIC50: 5.08E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196905(CHEMBL3906675)copy SMILEScopy InChI
Affinity DataIC50: 5.16E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196910(CHEMBL3943625)copy SMILEScopy InChI
Affinity DataIC50: 5.31E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196907(CHEMBL3904951)copy SMILEScopy InChI
Affinity DataIC50: 5.32E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196902(CHEMBL3931874)copy SMILEScopy InChI
Affinity DataIC50: 6.22E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VZDPubMed