Affinity DataKi: 0.0480nMAssay Description:Inhibitory activity against human adenosine A2A receptor expressed in HEK-293 cells by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against adenosine A2A receptor in rat striatal membranes by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C]-GR-218,231More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University of Milano/Bicocca
Curated by ChEMBL
University of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University of Milano/Bicocca
Curated by ChEMBL
University of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 184nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 342nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University of Milano/Bicocca
Curated by ChEMBL
University of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Inhibitory activity against human adenosine A1 receptor expressed in CHO cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 1.82E+3nMAssay Description:Displacement of [3H]-DPCPX from adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University of Milano/Bicocca
Curated by ChEMBL
University of Milano/Bicocca
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human adenosine A2B receptor expressed in HEK-293 cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against rat adenosine A3 receptor expressed in HEK-293 cells by displacement of [125I]-AB-MECAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 3.15E+4nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 3.28E+4nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 8.72E+4nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 1.27E+5nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
ETH Zurich
Curated by ChEMBL
ETH Zurich
Curated by ChEMBL
Affinity DataIC50: 2.91E+5nMAssay Description:Inhibition of bacterial InhA harboring S94A mutant using 2-trans-octenoyl-CoA or 2-trans-dodecenoyl-CoA as substrateMore data for this Ligand-Target Pair
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