Compile Data Set for Download or QSAR
Found 90 with Last Name = 'kissova' and Initial = 'm'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467697(CHEMBL4277981)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467700(CHEMBL4286927)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467698(CHEMBL4286320)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467694(CHEMBL4294817)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467696(CHEMBL4291408)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP484TPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467699(CHEMBL4278410)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467693(CHEMBL4288646)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467695(CHEMBL4283564)copy SMILEScopy InChI
Affinity DataKi:  74nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of recombinant full length N-terminal His6 tagged human FYN expressed in baculovirus infected sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467703(CHEMBL4281871)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant full length N-terminal His6 tagged human FYN expressed in baculovirus infected sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467702(CHEMBL4283149)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of LYN (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of LYN (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467701(CHEMBL4290337)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50142882(Butyl-[1-(2-chloro-2-phenyl-ethyl)-6-ethylsulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  320nMAssay Description:Inhibition of recombinant wild type c-ABL (unknown origin) after 5 mins by scintillation counting analysis in presence of [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1T4RPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230317(CHEMBL4091022)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230313(CHEMBL4068876)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230311(CHEMBL4063136)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50467704(CHEMBL4293733)copy SMILEScopy InChI
Affinity DataKi:  840nMAssay Description:Inhibition of human c-Src using KVEKIGEGTYGVVYK as substrate in presence of [gamma32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2S18PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50354489(CHEMBL1836680)copy SMILEScopy InChI
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of recombinant wild type c-ABL (unknown origin) after 5 mins by scintillation counting analysis in presence of [gamma32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1T4RPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230318(CHEMBL4103914)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230316(CHEMBL4088440)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230321(CHEMBL4073713)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230319(CHEMBL4060213)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230320(CHEMBL4100526)copy SMILEScopy InChI
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230312(CHEMBL4098763)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50230315(CHEMBL4096164)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged Src expressed in Sf21 cells using KVEKIGEGTYGVVYK as substrate after 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959KTBPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506077(CHEMBL4471507)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506070(CHEMBL4461468)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 20 mins in presence of [gamma-33P ATP] by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506070(CHEMBL4461468)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 5 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506062(CHEMBL4531023)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506060(CHEMBL4580215)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506064(CHEMBL4445768)copy SMILEScopy InChI
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506076(CHEMBL4447091)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506072(CHEMBL4590346)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 20 mins in presence of [gamma-33P ATP] by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506072(CHEMBL4590346)copy SMILEScopy InChI
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 5 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506073(CHEMBL4574818)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506072(CHEMBL4590346)copy SMILEScopy InChI
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 0 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506070(CHEMBL4461468)copy SMILEScopy InChI
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 0 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506065(CHEMBL4544312)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506069(CHEMBL4556068)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 0 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50206297(CHEMBL3911525)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant human Src using KVEKIGEGTYGVVYK as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP484TPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506061(CHEMBL4528964)copy SMILEScopy InChI
Affinity DataIC50: 4.84E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 5 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506071(CHEMBL4566690)copy SMILEScopy InChI
Affinity DataIC50: 5.21E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 20 mins in presence of [gamma-33P ATP] by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Universit£ degli Studi di Parma

Curated by ChEMBL
LigandPNGBDBM50506071(CHEMBL4566690)copy SMILEScopy InChI
Affinity DataIC50: 5.39E+3nMAssay Description:Inhibition of recombinant human full length His6-tagged PI4KIII beta expressed in Sf9 cells incubated for 0 mins in presence of [gamma-33P ATP] by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P92PWPubMed
Displayed 1 to 50 (of 90 total ) | Next | Last >>
Jump to: