Compile Data Set for Download or QSAR
Found 252 with Last Name = 'kuroha' and Initial = 'm'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50314948((S)-8-Acetyl-6,9-dihydroxy-3-methoxy-6b-methyl-1,7...)copy SMILEScopy InChI
Affinity DataKi:  82nMAssay Description:Binding affinity to PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9D21PubMed
TargetProtein kinase C-like 1(Candida albicans)
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of Candida albicans Pkc1 expressed in insect Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41R95PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600302(CHEMBL5193437)copy SMILES
Affinity DataIC50: 56nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600297(CHEMBL5174606)copy SMILES
Affinity DataIC50: 130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600297(CHEMBL5174606)copy SMILES
Affinity DataIC50: 130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600296(CHEMBL5177811)copy SMILES
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600300(CHEMBL5184238)copy SMILES
Affinity DataIC50: 170nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600298(CHEMBL5187549)copy SMILES
Affinity DataIC50: 190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600299(CHEMBL5191305)copy SMILES
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600304(CHEMBL5207535)copy SMILES
Affinity DataIC50: 260nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human PKCbeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41R95PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600297(CHEMBL5174606)copy SMILES
Affinity DataIC50: 380nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600297(CHEMBL5174606)copy SMILES
Affinity DataIC50: 380nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600300(CHEMBL5184238)copy SMILES
Affinity DataIC50: 420nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600302(CHEMBL5193437)copy SMILES
Affinity DataIC50: 460nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600295(CHEMBL5209027)copy SMILES
Affinity DataIC50: 610nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600296(CHEMBL5177811)copy SMILES
Affinity DataIC50: 610nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50314948((S)-8-Acetyl-6,9-dihydroxy-3-methoxy-6b-methyl-1,7...)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of PPARgamma assessed as transcriptional activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9D21PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600303(CHEMBL5180471)copy SMILES
Affinity DataIC50: 910nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600298(CHEMBL5187549)copy SMILES
Affinity DataIC50: 1.01E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human PKCalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41R95PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600304(CHEMBL5207535)copy SMILES
Affinity DataIC50: 1.03E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetCREB-binding protein(Homo sapiens (Human))TBA
LigandPNGBDBM50579801(CHEMBL5088992)copy SMILES
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CBP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600303(CHEMBL5180471)copy SMILES
Affinity DataIC50: 1.45E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600295(CHEMBL5209027)copy SMILES
Affinity DataIC50: 2.24E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579797(CHEMBL5071269)copy SMILES
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579796(CHEMBL5087034)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetCREB-binding protein(Homo sapiens (Human))TBA
LigandPNGBDBM50579798(CHEMBL5080324)copy SMILES
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of CBP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579801(CHEMBL5088992)copy SMILES
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600299(CHEMBL5191305)copy SMILES
Affinity DataIC50: 5.02E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human PKCgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41R95PubMed
TargetHistone acetyltransferase KAT7(Homo sapiens)TBA
LigandPNGBDBM50346552(CHEMBL1797936)copy SMILEScopy InChI
Affinity DataIC50: 7.81E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579799(CHEMBL5093074)copy SMILES
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579798(CHEMBL5080324)copy SMILES
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579800(CHEMBL5083461)copy SMILES
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50314950((S)-8-Acetyl-6,9-dihydroxy-3-methoxy-6b-methyl-1,7...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of PPARgamma assessed as transcriptional activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9D21PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579794(CHEMBL5086865)copy SMILES
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579795(CHEMBL5089215)copy SMILES
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase KAT6B(Homo sapiens)TBA
LigandPNGBDBM50346552(CHEMBL1797936)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50600297(CHEMBL5174606)copy SMILES
Affinity DataIC50: 2.50E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579792(CHEMBL5086573)copy SMILES
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579793(CHEMBL5074998)copy SMILES
Affinity DataIC50: 3.54E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))TBA
LigandPNGBDBM50346552(CHEMBL1797936)copy SMILEScopy InChI
Affinity DataIC50: 3.72E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50579791(CHEMBL5069865)copy SMILES
Affinity DataIC50: 3.73E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XQQPubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))TBA
LigandPNGBDBM50346552(CHEMBL1797936)copy SMILEScopy InChI
Affinity DataIC50: 3.89E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6H8TPubMed
Displayed 1 to 50 (of 252 total ) | Next | Last >>
Jump to: