Compile Data Set for Download or QSAR
Found 578 with Last Name = 'kusaka' and Initial = 'm'
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045514(CHEMBL3315315)copy SMILES
Affinity DataKi:  0.0260nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045510(CHEMBL3314227)copy SMILES
Affinity DataKi:  0.0270nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045500(CHEMBL3314217)copy SMILES
Affinity DataKi:  0.0280nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045509(CHEMBL3314226)copy SMILES
Affinity DataKi:  0.0340nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045513(Kisspeptin-10)copy SMILES
Affinity DataKi:  0.0350nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045499(CHEMBL3314216)copy SMILES
Affinity DataKi:  0.0360nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045507(CHEMBL3314224)copy SMILES
Affinity DataKi:  0.0360nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045498(CHEMBL3314215)copy SMILES
Affinity DataKi:  0.0370nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045512(CHEMBL3314229)copy SMILES
Affinity DataKi:  0.0380nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045506(CHEMBL3314223)copy SMILES
Affinity DataKi:  0.0390nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045517(CHEMBL3314209)copy SMILES
Affinity DataKi:  0.0520nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045507(CHEMBL3314224)copy SMILES
Affinity DataKi:  0.0690nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045515(CHEMBL3314207)copy SMILES
Affinity DataKi:  0.0740nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045498(CHEMBL3314215)copy SMILES
Affinity DataKi:  0.0770nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045516(CHEMBL3314208)copy SMILES
Affinity DataKi:  0.0860nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045512(CHEMBL3314229)copy SMILES
Affinity DataKi:  0.0870nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045509(CHEMBL3314226)copy SMILES
Affinity DataKi:  0.0870nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045513(Kisspeptin-10)copy SMILES
Affinity DataKi:  0.0880nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045511(CHEMBL3314228)copy SMILES
Affinity DataKi:  0.0890nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045518(CHEMBL3314213)copy SMILES
Affinity DataKi:  0.0960nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50442961(CHEMBL3086284)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045508(CHEMBL3314225)copy SMILES
Affinity DataKi:  0.110nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045505(CHEMBL3314222)copy SMILES
Affinity DataKi:  0.120nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045515(CHEMBL3314207)copy SMILES
Affinity DataKi:  0.130nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50442961(CHEMBL3086284)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045511(CHEMBL3314228)copy SMILES
Affinity DataKi:  0.170nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045501(CHEMBL3314218)copy SMILES
Affinity DataKi:  0.200nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045505(CHEMBL3314222)copy SMILES
Affinity DataKi:  0.830nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd.

Curated by ChEMBL
LigandPNGBDBM50045501(CHEMBL3314218)copy SMILES
Affinity DataKi:  3.60nMAssay Description:Displacement of radioligand from rat KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XSGPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50122654(1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)ami...)copy SMILEScopy InChI
Affinity DataIC50: 0.0600nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347985(CHEMBL1800156)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347996(CHEMBL1800663)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347996(CHEMBL1800663)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347986(CHEMBL1800155)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347989(CHEMBL1800668)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347982(CHEMBL1800159)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347984(CHEMBL1800157)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347997(CHEMBL1800661)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347997(CHEMBL1800661)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347994(CHEMBL1800666)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347987(CHEMBL1800153)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347989(CHEMBL1800668)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347995(CHEMBL1800664)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50122654(1-(4-(1-(2,6-difluorobenzyl)-5-((benzyl(methyl)ami...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM230879(US9346822, 41)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2251H2FUS Patent
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347983(CHEMBL1800158)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347986(CHEMBL1800155)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347987(CHEMBL1800153)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachadonic acid release using [5,6,8,9,11,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50348001(CHEMBL1800662)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]leuprorelin from recombinant human GnRH receptor expressed in CHO cells after 60 mins by X-ray counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N52MKPubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50347988(CHEMBL1800152 | US9346822, 40)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2251H2FUS Patent
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