Compile Data Set for Download or QSAR
Found 19 with Last Name = 'mezei' and Initial = 'm'
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189696(CHEMBL3827924)copy SMILEScopy InChI
Affinity DataKi:  4.80E+3nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189697(CHEMBL3827733)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189699(CHEMBL3827834)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189698(CHEMBL3827336)copy SMILEScopy InChI
Affinity DataKi:  1.69E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189711(CHEMBL3827805)copy SMILEScopy InChI
Affinity DataKi:  2.50E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189780(CHEMBL3827954)copy SMILEScopy InChI
Affinity DataKi:  3.31E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189762(CHEMBL3827451)copy SMILEScopy InChI
Affinity DataKi:  3.93E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells in presence of FITC-labeled SE...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054JTPubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50271179(2-(2-(quinolin-2-yl)vinyl)phenol | CHEMBL487942 | ...)copy SMILEScopy InChI
Affinity DataIC50: 4.63E+3nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50271178(1-(pyrrolidin-1-yl)-2-(quinoxalin-6-yl)ethanone | ...)copy SMILEScopy InChI
Affinity DataIC50: 5.83E+3nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50001270(2-(2-(quinolin-2-yl)vinyl)phenol | 2-(2-Quinolin-2...)copy SMILEScopy InChI
Affinity DataIC50: 6.42E+3nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50271180(2-(2-hydroxy-3-methoxystyryl)quinolin-8-ol | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 3.29E+4nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetEEF1AKMT4-ECE2 readthrough transcript protein(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50271181(2-(3-methoxystyryl)quinolin-8-ol | CHEMBL488140 | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.57E+4nMAssay Description:Reduction of recombinant ECE2 (unknown origin) activity measured by McaBk2 fluorescent substrate hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetNeprilysin(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50271178(1-(pyrrolidin-1-yl)-2-(quinoxalin-6-yl)ethanone | ...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Neprilysin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetNeprilysin(Homo sapiens (Human))
Mount Sinai School of Medicine

Curated by ChEMBL
LigandPNGBDBM50001270(2-(2-(quinolin-2-yl)vinyl)phenol | 2-(2-Quinolin-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Neprilysin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319VN5PubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189695(CHEMBL1198405)copy SMILEScopy InChI
Affinity DataKd:  2.38E+4nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells assessed as compound/protein/F...More data for this Ligand-Target Pair
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
TBA

Curated by ChEMBL
LigandPNGBDBM50476285(CHEMBL609729)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MG1PubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189780(CHEMBL3827954)copy SMILEScopy InChI
Affinity DataKd:  1.25E+5nMAssay Description:Binding affinity to CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells assessed as compound/protein/F...More data for this Ligand-Target Pair
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
TBA

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MG1PubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
Icahn School of Medicine at Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50189695(CHEMBL1198405)copy SMILEScopy InChI
Affinity DataKd:  5.00E+5nMAssay Description:Binding affinity to 15N-labeled CBX7ChD (7 to 66 residues) (unknown origin) expressed in RIPL-BL21 (DE3)-CodonPlus competent cells by HSQC/NMR titrat...More data for this Ligand-Target Pair