Affinity DataKi: 332nMAssay Description:Displacement of [3H]9cis-RA from human RXRalpha-LBD by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 384nMAssay Description:Displacement of NEt-C343 from human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as inhibition constant incubated for 2 hrs by...More data for this Ligand-Target Pair
Affinity DataKi: 391nMAssay Description:Displacement of NEt-C343 from human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as inhibition constant incubated for 2 hrs by...More data for this Ligand-Target Pair
Affinity DataKi: 425nMAssay Description:Displacement of [3H]9cis-RA from human RXRalpha-LBD by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Displacement of 6-(Ethyl-{5-isobutoxy-4-isopropyl-2-[(10-oxo-2,3,5,6-tetrahydro-1H,4H,10H-11-oxa-3a-aza-benzo[de]anthracene-9-carbonyl)-amino]-phenyl...More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2959N9FPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2959N9FPubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
Affinity DataKi: 3.16E+3nMAssay Description:Displacement of NEt-C343 from human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as inhibition constant incubated for 2 hrs by...More data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Displacement of NEt-C343 from human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as inhibition constant incubated for 2 hrs by...More data for this Ligand-Target Pair
Affinity DataKd: 705nMAssay Description:Binding affinity to human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as dissociated constant incubated for 2 hrs by tryptoph...More data for this Ligand-Target Pair
Affinity DataKd: 764nMAssay Description:Binding affinity to human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as dissociated constant incubated for 2 hrs by tryptoph...More data for this Ligand-Target Pair
Affinity DataKd: 277nMAssay Description:Binding affinity to human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as dissociated constant incubated for 2 hrs by tryptoph...More data for this Ligand-Target Pair
Affinity DataKd: 257nMAssay Description:Binding affinity to human RXRalpha-LBD by fluorescence binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to human RXRalpha-LBD assessed as binding constant from binding ratio at 327 nm by fluorometric titration assayMore data for this Ligand-Target Pair
Affinity DataKd: 281nMAssay Description:Binding affinity to human RXRalpha-LBD expressed in African green monkey COS-1 cells assessed as dissociated constant incubated for 2 hrs by tryptoph...More data for this Ligand-Target Pair
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