Compile Data Set for Download or QSAR
Found 111 with Last Name = 'payton' and Initial = 'm'
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326208(4-(4-Fluorophenyl)-N-(4-(3-(2-(methylamino)pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326204(CHEMBL1243137 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326207(CHEMBL1243294 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50557717(CHEMBL4743666)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404039(CHEMBL5289941)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326202(CHEMBL1243042 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404036(CHEMBL5076091)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326198(CHEMBL1242977 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Mus musculus)TBA
LigandPNGBDBM50404035(CHEMBL5287177)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404000(CHEMBL5279604)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404034(CHEMBL5077043)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404037(CHEMBL5287302)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403677(CHEMBL5288088)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404035(CHEMBL5287177)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of pig brain farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326205(CHEMBL1243167 | N-(2-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404033(CHEMBL5083562)copy SMILEScopy InChI
Affinity DataIC50: 135nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404030(CHEMBL5278809)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403999(CHEMBL5276902)copy SMILEScopy InChI
Affinity DataIC50: 165nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50404031(CHEMBL5270982)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326203(CHEMBL1243073 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403678(CHEMBL5276935)copy SMILEScopy InChI
Affinity DataIC50: 253nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403675(CHEMBL5081638)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326201(4-Chloro-N-(3-methyl-4-(3-(2-(methylamino)pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 335nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403676(CHEMBL5284647)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326198(CHEMBL1242977 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 385nMAssay Description:Inhibition of LCK by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403557(CHEMBL5084830)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326200(3-Chloro-N-(3-methyl-4-(3-(2-(methylamino)pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326198(CHEMBL1242977 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 503nMAssay Description:Inhibition of Abl by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403553(CHEMBL5266739)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326209(CHEMBL1243108 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 542nMAssay Description:Inhibition of Aurora B by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403674(CHEMBL5083490)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Rabbit pulmonary artery(RPA) assay.More data for this Ligand-Target Pair
In DepthDetails
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326198(CHEMBL1242977 | N-(3-Methyl-4-(3-(2-(methylamino)p...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of Tie-2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PLK1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p70s6k by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of JNK2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of BTK by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Jak3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK5 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Zap70 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of IGFR1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EphB4 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EGFR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of c-Met by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Erk1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKBalpha by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50326206(CHEMBL1243200 | N-(4-(3-(2-(Methylamino)pyrimidin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Jak2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C829H0PubMed
TargetKinesin-like protein KIF18A(Homo sapiens)TBA
LigandPNGBDBM50403556(CHEMBL5287687)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+3nMAssay Description:Antagonist activity against Tachykinin receptor 2 was measured by Hamster isolated trachea(HT) assay.More data for this Ligand-Target Pair
In DepthDetails
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