Affinity DataKi: 5.80nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn
Curated by ChEMBL
University of Bonn
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn
Curated by ChEMBL
University of Bonn
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn
Curated by ChEMBL
University of Bonn
Curated by ChEMBL
Affinity DataKi: 1.56E+3nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.64E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn
Curated by ChEMBL
University of Bonn
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.86E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 1.98E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.15E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.26E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.45E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.52E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.55E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 2.92E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 4.43E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 4.49E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 5.02E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 5.56E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 5.65E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 5.72E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 5.73E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.76E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 6.28E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.40E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 6.77E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 6.81E+3nMAssay Description:Inhibition of human TGase 2 using R-I-Cad/DMC as substrate preincubated for 5 mins followed by substrate addition measured at 30 secs interval over 9...More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.12E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.32E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.55E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.71E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf
Curated by ChEMBL
Affinity DataKi: 7.76E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair