Compile Data Set for Download or QSAR
Found 159 with Last Name = 'pietsch' and Initial = 'm'
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084235(2-Diethylamino-benzo[4,5]thieno[2,3-d][1,3]oxazin-...)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084232(2-(diethylamino)-5-isopropyl-4H-thieno[2,3-d][1,3]...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084233(2-Diethylamino-6,7-dihydro-5H-cyclopenta[4,5]thien...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50064308(2-Diethylamino-5,6,7,8-tetrahydro-benzo[4,5]thieno...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084234(2-Diethylamino-6,7,8,9-tetrahydro-5H-3-oxa-10-thia...)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084227(2-(diethylamino)-5-methyl-4-oxo-4H-thieno[2,3-d][1...)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084230(2-Diethylamino-thieno[3,2-d][1,3]oxazin-4-one | CH...)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084229(2-Diethylamino-5-methyl-5,6,7,8-tetrahydro-benzo[4...)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084236(2-Diethylamino-thieno[2,3-d][1,3]oxazin-4-one | CH...)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084231(2-Diethylamino-benzo[d][1,3]oxazin-4-one | CHEMBL3...)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University of Leipzig

Curated by ChEMBL
LigandPNGBDBM50084228(2-(diethylamino)-5-methyl-4H-thieno[2,3-d][1,3]oxa...)copy SMILEScopy InChI
Affinity DataKi:  450nMAssay Description:Inhibitory activity of the compound was tested against human leukocyte elastaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936RGPubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084233(2-Diethylamino-6,7-dihydro-5H-cyclopenta[4,5]thien...)copy SMILEScopy InChI
Affinity DataKi:  580nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179322(6,7-dihydro-2-(dimethylamino)-4H,5H-cyclopenta[4,5...)copy SMILEScopy InChI
Affinity DataKi:  630nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179314(5,6,7,8-tetrahydro-2-(dimethylamino)-7-(2-methyl-p...)copy SMILEScopy InChI
Affinity DataKi:  660nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)copy SMILEScopy InChI
Affinity DataKi:  1.56E+3nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084229(2-Diethylamino-5-methyl-5,6,7,8-tetrahydro-benzo[4...)copy SMILEScopy InChI
Affinity DataKi:  1.64E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179312(7-benzyl-5,6,7,8-tetrahydro-2-(dimethylamino)-4H-p...)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity AChE from Electrophorus electricus using ATCh substrate and DTNB by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50064308(2-Diethylamino-5,6,7,8-tetrahydro-benzo[4,5]thieno...)copy SMILEScopy InChI
Affinity DataKi:  1.86E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461625(CHEMBL4228924)copy SMILEScopy InChI
Affinity DataKi:  1.98E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179331(5,6,7,8-tetrahydro-2-(dimethylamino)-4H-benzo[4,5]...)copy SMILEScopy InChI
Affinity DataKi:  2.15E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461612(CHEMBL4227301)copy SMILEScopy InChI
Affinity DataKi:  2.26E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461615(CHEMBL4228875)copy SMILEScopy InChI
Affinity DataKi:  2.45E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461619(CHEMBL4224727)copy SMILEScopy InChI
Affinity DataKi:  2.52E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461617(CHEMBL4229073)copy SMILEScopy InChI
Affinity DataKi:  2.55E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461633(CHEMBL4227896)copy SMILEScopy InChI
Affinity DataKi:  2.60E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461610(CHEMBL4227835)copy SMILEScopy InChI
Affinity DataKi:  2.92E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461626(CHEMBL4228542)copy SMILEScopy InChI
Affinity DataKi:  3.50E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179326(2-(diethylamino)-5,6-dimethyl-4H-thieno[2,3-d][1,3...)copy SMILEScopy InChI
Affinity DataKi:  4.30E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461609(CHEMBL4227328)copy SMILEScopy InChI
Affinity DataKi:  4.43E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461621(CHEMBL4226871)copy SMILEScopy InChI
Affinity DataKi:  4.49E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461622(CHEMBL4228726)copy SMILEScopy InChI
Affinity DataKi:  5.02E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461620(CHEMBL4228541)copy SMILEScopy InChI
Affinity DataKi:  5.56E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461608(CHEMBL4228671)copy SMILEScopy InChI
Affinity DataKi:  5.65E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179329(2-morpholin-4-yl-5,6,7,8-tetrahydro-benzo[4,5]thie...)copy SMILEScopy InChI
Affinity DataKi:  5.70E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461635(CHEMBL4228810)copy SMILEScopy InChI
Affinity DataKi:  5.72E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50400621(CHEMBL2203451)copy SMILEScopy InChI
Affinity DataKi:  5.73E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50179318(2-dimethylamino-5,8-dihydro-4H,6H-thiopyrano[4',3'...)copy SMILEScopy InChI
Affinity DataKi:  5.76E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084234(2-Diethylamino-6,7,8,9-tetrahydro-5H-3-oxa-10-thia...)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461607(CHEMBL4228168)copy SMILEScopy InChI
Affinity DataKi:  6.28E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084232(2-(diethylamino)-5-isopropyl-4H-thieno[2,3-d][1,3]...)copy SMILEScopy InChI
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461630(CHEMBL4225325)copy SMILEScopy InChI
Affinity DataKi:  6.77E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461614(CHEMBL4226594)copy SMILEScopy InChI
Affinity DataKi:  6.81E+3nMAssay Description:Inhibition of human TGase 2 using R-I-Cad/DMC as substrate preincubated for 5 mins followed by substrate addition measured at 30 secs interval over 9...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461616(CHEMBL4224787)copy SMILEScopy InChI
Affinity DataKi:  7.12E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461629(CHEMBL4228146)copy SMILEScopy InChI
Affinity DataKi:  7.32E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetBile salt-activated lipase(Bos taurus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50084235(2-Diethylamino-benzo[4,5]thieno[2,3-d][1,3]oxazin-...)copy SMILEScopy InChI
Affinity DataKi:  7.50E+3nMAssay Description:Inhibitory activity against bovine pancreatic CEase in presence of pNPB chromogenic substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6XB4PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461618(CHEMBL4225321)copy SMILEScopy InChI
Affinity DataKi:  7.55E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461636(CHEMBL4228357)copy SMILEScopy InChI
Affinity DataKi:  7.60E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461624(CHEMBL4226385)copy SMILEScopy InChI
Affinity DataKi:  7.71E+3nMAssay Description:Irreversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Helmholtz-Zentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50461611(CHEMBL4226785)copy SMILEScopy InChI
Affinity DataKi:  7.76E+3nMAssay Description:Reversible inhibition of human TGase 2 using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66PC7PubMed
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