Compile Data Set for Download or QSAR
Found 3 with Last Name = 'ponelle' and Initial = 'm'
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Novartis Institutes for BioMedical Research and Novartis Pharma Development

Curated by ChEMBL
LigandPNGBDBM50030448(8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN | CHEMBL269732 ...)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:Inhibitory activity against macrophilin (FKBP-12)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N81WKPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Novartis Institutes for BioMedical Research and Novartis Pharma Development

Curated by ChEMBL
LigandPNGBDBM50153090(CHEMBL411735 | Macrolide derivative)copy SMILEScopy InChI
Affinity DataIC50: 1.45nMAssay Description:Inhibitory activity against macrophilin (FKBP-12)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N81WKPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Novartis Institutes for BioMedical Research and Novartis Pharma Development

Curated by ChEMBL
LigandPNGBDBM50153091(CHEMBL265123 | Macrolide derivative)copy SMILEScopy InChI
Affinity DataIC50: 1.88nMAssay Description:Inhibitory activity against macrophilin (FKBP-12)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N81WKPubMed