Compile Data Set for Download or QSAR
Found 162 with Last Name = 'schiedel' and Initial = 'm'
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148829(CHEMBL3769432)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human SIRT2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Inhibition of recombinant His-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human CREBBP by AlphaScreen assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50459845(CHEMBL4227437)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50459842(CHEMBL4228286)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273645(CHEMBL4129171)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273645(CHEMBL4129171)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273654(CHEMBL4127935)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273654(CHEMBL4127935)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148782(CHEMBL3770049)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148782(CHEMBL3770049)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B33Z7PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148789(CHEMBL3771286)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant His-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follow...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273629(CHEMBL4128951)copy SMILEScopy InChI
Affinity DataIC50: 234nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273629(CHEMBL4128951)copy SMILEScopy InChI
Affinity DataIC50: 235nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50459841(CHEMBL4225467)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B33Z7PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148784(CHEMBL3769991)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273652(CHEMBL4130228)copy SMILEScopy InChI
Affinity DataIC50: 269nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273652(CHEMBL4130228)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273619(CHEMBL4125731)copy SMILEScopy InChI
Affinity DataIC50: 295nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273619(CHEMBL4125731)copy SMILEScopy InChI
Affinity DataIC50: 296nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273650(CHEMBL4127775)copy SMILEScopy InChI
Affinity DataIC50: 302nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273650(CHEMBL4127775)copy SMILEScopy InChI
Affinity DataIC50: 303nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50459843(CHEMBL4225505)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B33Z7PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148791(CHEMBL3770797)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50151661(CHEMBL3752296)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of human CREBBPMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148792(CHEMBL3771296)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50151661(CHEMBL3752296)copy SMILEScopy InChI
Affinity DataIC50: 323nMAssay Description:Inhibition of CREBBP (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273626(CHEMBL4126542)copy SMILEScopy InChI
Affinity DataIC50: 377nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273649(CHEMBL2335143)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273626(CHEMBL4126542)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273649(CHEMBL2335143)copy SMILEScopy InChI
Affinity DataIC50: 384nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148783(CHEMBL3771164)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148781(CHEMBL3770903)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of recombinant human His10-tagged Sirt2 (56 to 356 residues) expressed in Escherichia coli BL21(DE3) using Z-(Ac)Lys-AMC as substrate meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148781(CHEMBL3770903)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273643(CHEMBL4126957)copy SMILEScopy InChI
Affinity DataIC50: 478nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273643(CHEMBL4126957)copy SMILEScopy InChI
Affinity DataIC50: 479nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148793(CHEMBL3770258)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273646(CHEMBL4126698)copy SMILEScopy InChI
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273646(CHEMBL4126698)copy SMILEScopy InChI
Affinity DataIC50: 495nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148794(CHEMBL3771278)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Albert-Ludwigs-University Freiburg

Curated by ChEMBL
LigandPNGBDBM50148795(CHEMBL3769999)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of N-terminal his6-tagged human SIRT2 (25 to 389 amino acids) using ZMAL as substrate after 4 hrs by fluorescence-based microplate reader ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1FH2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273687(CHEMBL4129017)copy SMILEScopy InChI
Affinity DataIC50: 585nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273687(CHEMBL4129017)copy SMILEScopy InChI
Affinity DataIC50: 589nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273655(CHEMBL4128749)copy SMILEScopy InChI
Affinity DataIC50: 603nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273655(CHEMBL4128749)copy SMILEScopy InChI
Affinity DataIC50: 604nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273616(CHEMBL4128199)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273616(CHEMBL4128199)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273651(CHEMBL4126757)copy SMILEScopy InChI
Affinity DataIC50: 722nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273651(CHEMBL4126757)copy SMILEScopy InChI
Affinity DataIC50: 724nMAssay Description:Inhibition of recombinant His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells preincubated for 30 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89FXZPubMed
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