Compile Data Set for Download or QSAR
Found 40 with Last Name = 'skingle' and Initial = 'm'
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  0.126nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469879(CHEMBL72088)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469882(CHEMBL73446)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469881(CHEMBL311150)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469875(CHEMBL72981)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50469881(CHEMBL311150)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469878(CHEMBL72700)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469876(CHEMBL306384)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50469876(CHEMBL306384)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1B receptor in rat striatal membrane with [125I]- iodocyanopindololMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469877(CHEMBL72092)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor in guinea-pig striatum in presence of BMY-7378 and mesulergineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469881(CHEMBL311150)copy SMILEScopy InChI
Affinity DataKi:  251nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus with [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 2C(PIG)
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against alpha-2 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against alpha-1 adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity against muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469875(CHEMBL72981)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus with [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469876(CHEMBL306384)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469878(CHEMBL72700)copy SMILEScopy InChI
Affinity DataKi:  5.01E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  6.31E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi:  6.31E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469880(CHEMBL75771)copy SMILEScopy InChI
Affinity DataKi:  6.31E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Tested for 5-hydroxytryptamine receptor uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Glaxo Research and Development Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM79215(CHEMBL15928 | GR 127935 | GR 127935 hydrochloride ...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58JX0PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50469877(CHEMBL72092)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Research and Development Ltd.

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat hippocampus using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29889QBPubMed