Compile Data Set for Download or QSAR
Found 183 with Last Name = 'yamasaki' and Initial = 'm'
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289647(CHEMBL263855 | Compound RES-701-1(1-10)/[A15]ET-1)copy SMILEScopy InChI
Affinity DataIC50: 0.240nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081F2
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460089(CHEMBL4226373)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289650(CHEMBL414047 | Compound RES-701-1(1-10)/[A15]ET-3)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081F2
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452856(CHEMBL4217811)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452853(CHEMBL4087736)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452850(CHEMBL4203255)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452854(CHEMBL4205112)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460093(CHEMBL4226313)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289648(CHEMBL408437 | Compound RES-701-1(1-10)/[A15]SRTX6...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081F2
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452843(CHEMBL4217478)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460088(CHEMBL4225541)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452840(CHEMBL4209940)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452846(CHEMBL4205579)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452848(CHEMBL4213410)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452839(CHEMBL4210540)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460097(CHEMBL4228650)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460074(CHEMBL4228907)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460089(CHEMBL4226373)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at RORgammat (unknown origin) expressed in human Jurkat cells assessed as inhibition of transcriptional activity after overn...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452847(CHEMBL4206093)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452842(CHEMBL4210727)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460082(CHEMBL4227433)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452847(CHEMBL4206093)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inverse agonist activity at RORgammat in human Jurkat cells assessed as inhibition of transcriptional activity after overnight incubation by human IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289112(CHEMBL438745 | RES-701-1-C-terminal analogue)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182G7
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452844(CHEMBL4214337)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452850(CHEMBL4203255)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inverse agonist activity at RORgammat in human Jurkat cells assessed as inhibition of transcriptional activity after overnight incubation by human IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460074(CHEMBL4228907)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Inverse agonist activity at RORgammat (unknown origin) expressed in human Jurkat cells assessed as inhibition of transcriptional activity after overn...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289108(CHEMBL384792 | RES-701-1 | RES-701-1-C-terminal an...)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182G7
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460075(CHEMBL4225105)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452852(CHEMBL4210449)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460080(CHEMBL4224762)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452841(CHEMBL4205062)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452849(CHEMBL4213861)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Displacement of BODIPY-labeled ligand from human His-tagged RORgammat after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277598(CHEMBL453211 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2V1GPubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277599(CHEMBL507541 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2V1GPubMed
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289111(CHEMBL411057 | RES-701-1-C-terminal analogue)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182G7
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289108(CHEMBL384792 | RES-701-1 | RES-701-1-C-terminal an...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Binding activity to ET-B receptor on bovine cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081F2
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inverse agonist activity at RORgammat (unknown origin) expressed in human Jurkat cells assessed as inhibition of transcriptional activity after overn...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inverse agonist activity at RORgammat (unknown origin) expressed in human Jurkat cells assessed as inhibition of transcriptional activity after overn...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetEndothelin receptor type B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289107(CHEMBL263294 | RES-701-1-C-terminal analogue)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding activity against Endothelin B receptor expressed from bovine cerebellum membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182G7
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50458200(CHEMBL3314031)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at RORgammat (unknown origin) expressed in human Jurkat cells assessed as inhibition of transcriptional activity after overn...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277597(CHEMBL501242 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2V1GPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452848(CHEMBL4213410)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at RORgammat in human Jurkat cells assessed as inhibition of transcriptional activity after overnight incubation by human IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67KH2PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460090(CHEMBL4225984)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50452848(CHEMBL4213410)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at RORgammat in human Jurkat cells assessed as inhibition of transcriptional activity after overnight incubation by human IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ71BRPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50460083(CHEMBL4224797)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of BODIPY-labeled-(R)-N-(2-(3,5-difluoro-4-(trimethylsilyl)phenylamino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-5-(2-((1-(difluoroboryl)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R7JPubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277595(CHEMBL445281 | N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2V1GPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50454142(CHEMBL4214211)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inverse agonist activity at RORgammat in human Jurkat cells assessed as inhibition of transcriptional activity after overnight incubation by human IL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67KH2PubMed
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