TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK5/p35 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK2/CyclinE (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 465nMAssay Description:Inhibition of IKKbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 911nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LRRK2 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ITK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of IKKbeta (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAPK14 (unknown origin) after 22 mins by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRKA (unknown origin)More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK3 (unknown origin) after 22 mins by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PAK1 (unknown origin)More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Eppley Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC2 expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange ac...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC2 expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange ac...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Institute for Research in Cancer and Allied Diseases
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
Affinity DataKd: 1.07E+3nMAssay Description:Binding affinity to CDK9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 385nMAssay Description:Binding affinity to CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 135nMAssay Description:Binding affinity to CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 815nMAssay Description:Binding affinity to CDK5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Binding affinity to CDK5 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.06E+3nMAssay Description:Binding affinity to CDK9 (unknown origin)More data for this Ligand-Target Pair