Compile Data Set for Download or QSAR
Found 124 with Last Name = 'van volkenburg' and Initial = 'm'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50140541((S)-2-Amino-2-cyclohexyl-1-(3,3-difluoro-pyrrolidi...)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50140527((S)-2-Amino-2-cyclohexyl-1-((S)-3-fluoro-pyrrolidi...)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172141((S)-2-Amino-2-cyclohexyl-1-(3,4-difluoro-pyrrolidi...)copy SMILEScopy InChI
Affinity DataKi:  61nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV calculated from IC50 from standard dose inhibition curve using cheng-Prussoff equation; range=61+/...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172144((S)-2-Amino-2-cyclohexyl-1-(2,3,4,5-tetrafluoro-py...)copy SMILEScopy InChI
Affinity DataKi:  81nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172143((S)-2-Amino-2-cyclohexyl-1-(3-fluoro-azetidin-1-yl...)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172139((S)-2-Amino-2-cyclohexyl-1-(3,3-difluoro-azetidin-...)copy SMILEScopy InChI
Affinity DataKi:  117nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM12191((2S)-2-amino-2-cyclohexyl-1-(pyrrolidin-1-yl)ethan...)copy SMILEScopy InChI
Affinity DataKi:  121nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50140539((S)-2-Amino-2-cyclohexyl-1-((R)-3-fluoro-pyrrolidi...)copy SMILEScopy InChI
Affinity DataKi:  128nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172145((S)-2-Amino-2-cyclohexyl-1-((3R,4R)-3,4-difluoro-p...)copy SMILEScopy InChI
Affinity DataKi:  504nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172140((S)-2-Amino-2-cyclohexyl-1-((3S,4S)-3,4-difluoro-p...)copy SMILEScopy InChI
Affinity DataKi:  1.27E+3nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50172142((S)-2-Amino-1-azetidin-1-yl-2-cyclohexyl-ethanone ...)copy SMILEScopy InChI
Affinity DataKi:  3.35E+3nMAssay Description:Inhibitory constant against Dipeptidylpeptidase IV activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K78M0PubMed
LigandPNGBDBM50390333(CHEMBL2070733)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390334(CHEMBL2070735)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390332(CHEMBL2070732)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390334(CHEMBL2070735)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PDE8AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390373(CHEMBL2070914)copy SMILEScopy InChI
Affinity DataIC50: 3.63nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390335(CHEMBL2070736)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390366(CHEMBL2070935)copy SMILEScopy InChI
Affinity DataIC50: 6.79nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390324(CHEMBL2070604)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390313(CHEMBL2070595)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390352(CHEMBL2070901)copy SMILEScopy InChI
Affinity DataIC50: 12.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390367(CHEMBL2070907)copy SMILEScopy InChI
Affinity DataIC50: 13.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390308(CHEMBL2070592)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390309(CHEMBL2070591)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390371(CHEMBL2070912)copy SMILEScopy InChI
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390378(CHEMBL2070919)copy SMILEScopy InChI
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390339(CHEMBL2070769)copy SMILEScopy InChI
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390363(CHEMBL2070932)copy SMILEScopy InChI
Affinity DataIC50: 17.7nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390336(CHEMBL2070737)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390364(CHEMBL2070933)copy SMILEScopy InChI
Affinity DataIC50: 21.4nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390343(CHEMBL2070773)copy SMILEScopy InChI
Affinity DataIC50: 21.6nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390329(CHEMBL2070729)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390338(CHEMBL2070734)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390320(CHEMBL2070600)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390375(CHEMBL2070916)copy SMILEScopy InChI
Affinity DataIC50: 25.5nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390384(CHEMBL2070925)copy SMILEScopy InChI
Affinity DataIC50: 31.5nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390379(CHEMBL2070920)copy SMILEScopy InChI
Affinity DataIC50: 31.7nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390358(CHEMBL2070927)copy SMILEScopy InChI
Affinity DataIC50: 38.8nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390306(CHEMBL2070768)copy SMILEScopy InChI
Affinity DataIC50: 39.2nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390331(CHEMBL2070731)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390381(CHEMBL2070922)copy SMILEScopy InChI
Affinity DataIC50: 43.9nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390312(CHEMBL2070594)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390357(CHEMBL2070926)copy SMILEScopy InChI
Affinity DataIC50: 48.4nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390380(CHEMBL2070921)copy SMILEScopy InChI
Affinity DataIC50: 52.4nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390365(CHEMBL2070934)copy SMILEScopy InChI
Affinity DataIC50: 53.8nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390376(CHEMBL2070917)copy SMILEScopy InChI
Affinity DataIC50: 55.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390350(CHEMBL2070899)copy SMILEScopy InChI
Affinity DataIC50: 61.2nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390340(CHEMBL2070770)copy SMILEScopy InChI
Affinity DataIC50: 70.7nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390349(CHEMBL2070898)copy SMILEScopy InChI
Affinity DataIC50: 72.7nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
LigandPNGBDBM50390382(CHEMBL2070923)copy SMILEScopy InChI
Affinity DataIC50: 74.6nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67J0XPubMed
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