Compile Data Set for Download or QSAR
Found 376 with Last Name = 'carnerup' and Initial = 'ma'
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539844(CHEMBL4643061)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560311(CHEMBL4756197)copy SMILES
Affinity DataIC50: 1nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of N-terminal His-tagged human JAK3 catalytic domain incubated for 20 mins in presence of TK substrate-biotin by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536220(CHEMBL4528395)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560315(CHEMBL4763360)copy SMILES
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560326(CHEMBL4758563)copy SMILES
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560313(CHEMBL4762028)copy SMILES
Affinity DataIC50: 2nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539841(CHEMBL4639606)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536209(CHEMBL4539949)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536208(CHEMBL4483364)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536217(CHEMBL4517645)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of N-terminal His-tagged human JAK2 catalytic domain incubated for 20 mins in presence of TK substrate-biotin by TR-FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539840(CHEMBL4649484)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536198(CHEMBL4534573)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536221(CHEMBL4554460)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536214(CHEMBL4560212)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536200(CHEMBL4483513)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539842(CHEMBL4636507)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536209(CHEMBL4539949)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536197(CHEMBL4521312)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536216(CHEMBL4580425)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536215(CHEMBL4569613)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536208(CHEMBL4483364)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536198(CHEMBL4534573)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536208(CHEMBL4483364)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536204(CHEMBL4563039)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM159748(US10966980, Example 2 | US9035074, 2)copy SMILES
Affinity DataIC50: 5.10nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536200(CHEMBL4483513)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536205(CHEMBL4543715)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536198(CHEMBL4534573)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539831(CHEMBL4639973)copy SMILEScopy InChI
Affinity DataIC50: 6.40nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536217(CHEMBL4517645)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560319(CHEMBL4759758)copy SMILES
Affinity DataIC50: 7nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560323(CHEMBL4777937)copy SMILES
Affinity DataIC50: 7nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536217(CHEMBL4517645)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536209(CHEMBL4539949)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536222(CHEMBL4531121)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536214(CHEMBL4560212)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536218(CHEMBL4516561)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536212(CHEMBL4551061)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560317(CHEMBL4795123)copy SMILES
Affinity DataIC50: 8nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50560324(CHEMBL4755015)copy SMILES
Affinity DataIC50: 9nMAssay Description:Agonist activity at human glucocorticoid receptor in PBMC assessed as inhibition of LPS-induced TNFalpha releaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5XPNPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536221(CHEMBL4554460)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536215(CHEMBL4569613)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Inhibition of human Gst-tagged JAK1 (850 to 1154 residues) expressed in baculovirus using biotin-synthetic peptide as substrate after 40 mins by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536218(CHEMBL4516561)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human His-tagged JAK3 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536222(CHEMBL4531121)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536221(CHEMBL4554460)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50536200(CHEMBL4483513)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human His-tagged JAK2 expressed in baculovirus using biotin-synthetic peptide as substrate after 20 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC146JPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
GVK Biosciences Private Limited

Curated by ChEMBL
LigandPNGBDBM50539839(CHEMBL4638030)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal GST-tagged human JAK1 catalytic domain (850 to 1154 residues) incubated for 40 mins in presence of TK substrate-biotin by TR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V08PubMed
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