Compile Data Set for Download or QSAR
Found 645 with Last Name = 'flynn' and Initial = 'ma'
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077930(5-{5-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-metho...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077933(4-{5-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-metho...)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057169(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077934(3-Benzo[1,3]dioxol-5-yl-4-[3,4-dimethoxy-5-(2-morp...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077935(CHEMBL308646 | {5-[4-Benzo[1,3]dioxol-5-yl-2-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077936(4-{5-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-metho...)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034267(3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034267(3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077946(5-{5-[4-Benzo[1,3]dioxol-5-yl-2-hydroxy-2-(4-metho...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057164(CHEMBL10862 | Sodium; (Z)-2-(7-methoxy-benzo[1,3]d...)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290981(CHEMBL319452 | PD-163140 | [4-Benzo[1,3]dioxol-5-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034267(3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...)copy SMILEScopy InChI
Affinity DataIC50: 0.370nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077944(CHEMBL408055 | Sodium; 3-{5-[4-benzo[1,3]dioxol-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290983(3-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057150(5-Hydroxy-3-(7-methoxy-benzo[1,3]dioxol-5-yl)-5-(4...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057202(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-3-m...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290980(2-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290984(2-[4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077941(3-Benzo[1,3]dioxol-5-yl-4-[3,4-dimethoxy-5-(3-morp...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057178(CHEMBL10847 | Sodium; (Z)-2-(7-methoxy-benzo[1,3]d...)copy SMILEScopy InChI
Affinity DataIC50: 0.780nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290982(Allyl-carbamic acid 4-benzo[1,3]dioxol-5-yl-2-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057189(5-Hydroxy-3-(7-methoxy-benzo[1,3]dioxol-5-yl)-5-(4...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057166(CHEMBL10922 | Sodium; (Z)-2-benzo[1,3]dioxol-5-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.980nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077943(3-Benzo[1,3]dioxol-5-yl-4-[3-(3-dimethylamino-prop...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034267(3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057153(CHEMBL10832 | Sodium; (Z)-2-benzo[1,3]dioxol-5-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286614(CHEMBL155943 | CHEMBL3143473 | Sodium; 2-[2-{2-[(2...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against endothelin B (ETB) receptor using human girardi heart cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081DM
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057154(CHEMBL10697 | N-{4-[4-Benzo[1,3]dioxol-5-yl-2-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057179(3-Benzo[1,3]dioxol-5-yl-4-(3,4-dimethoxy-benzyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057181(3-Benzo[1,3]dioxol-5-yl-4-(3,5-dimethoxy-benzyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057167(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034259(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-4-(4-methoxy-ben...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077938(3-Benzo[1,3]dioxol-5-yl-4-{3,4-dimethoxy-5-[3-(4-m...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287200(1-Benzo[1,3]dioxol-5-ylmethyl-5,6-dimethoxy-3-(3,4...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35TMT
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290979(((S)-1-Naphthalen-1-yl-ethyl)-carbamic acid 4-benz...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077947(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50290979(((S)-1-Naphthalen-1-yl-ethyl)-carbamic acid 4-benz...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity for human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8584G
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057194(3-Benzo[1,3]dioxol-5-yl-4-(2,5-dimethoxy-benzyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50034269(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-4-(4-methoxy-3-m...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077945(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-dimethylamino-etho...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057192(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-4-(3-methoxy-ben...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032181(2-{1-[1-(2-carboxy-1-{1-[10,11-dihydro-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057207(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032175((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50077942(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-(4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of [125I]-ET-1 binding to recombinant human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12404PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057160(3-Benzo[1,3]dioxol-5-yl-5-hydroxy-4-(4-methanesulf...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Binding affinity against human cloned endothelin A receptor expressed in LTK-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287200(1-Benzo[1,3]dioxol-5-ylmethyl-5,6-dimethoxy-3-(3,4...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35TMT
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032181(2-{1-[1-(2-carboxy-1-{1-[10,11-dihydro-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50057213(CHEMBL10905 | Potassium; (Z)-3-(4-acetylamino-benz...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of Endothelin A receptor mediated (ET-1) release of arachidonic acid from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8XG5PubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287183(1-Benzo[1,3]dioxol-5-ylmethyl-3-(benzo[1,3]dioxol-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35TMT
Displayed 1 to 50 (of 645 total ) | Next | Last >>
Jump to: