Affinity DataIC50: 2nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 144nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: 205nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:In vitro binding affinity of the compound against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in human CYP3A4 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 235nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 253nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
Affinity DataIC50: 272nMAssay Description:Inhibition of binding to ER in Ad5-wt-ER-infected HAECT1 cells by NFkappaB-mediated luciferase reporterMore data for this Ligand-Target Pair
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