Compile Data Set for Download or QSAR
Found 230 with Last Name = 'singh' and Initial = 'mp'
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240209(CHEMBL4068526)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240227(CHEMBL4084391)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity was determined against HSV-1 Ribonucleoside diphosphate reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240213(CHEMBL4085366)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240224(CHEMBL4095856)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50228080(2',15'-dimethyl-5,5'-dioxo-(9'R)-spiro[tetrahydrof...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at mineralocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by ...More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240216(CHEMBL4074076)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240226(CHEMBL4065459)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HSV-1 Ribonucleoside diphosphate reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at glucocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at estrogen receptor beta ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381517(CHEMBL2017748)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240218(CHEMBL4059858)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at estrogen receptor alpha ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Displacement of progesterone from progesterone receptor in human T47D cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381530(CHEMBL2017761)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240227(CHEMBL4084391)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibitory activity was determined against HSV-1 Ribonucleoside diphosphate reductaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240219(CHEMBL4100838)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381510(CHEMBL2017741)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240204(CHEMBL4081527)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against HSV-1 Ribonucleoside diphosphate reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Integral BioSciences, Pvt. Ltd.

Curated by ChEMBL
LigandPNGBDBM50201721(CHEMBL3964073)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918G5PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240217(CHEMBL4063659)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381513(CHEMBL2017744)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Integral BioSciences, Pvt. Ltd.

Curated by ChEMBL
LigandPNGBDBM50201721(CHEMBL3964073)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918G5PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240211(CHEMBL4104586)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381513(CHEMBL2017744)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381510(CHEMBL2017741)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381511(CHEMBL2017742)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381527(CHEMBL2017757)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381531(CHEMBL2017762)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381512(CHEMBL2017743)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
Integral BioSciences, Pvt. Ltd.

Curated by ChEMBL
LigandPNGBDBM350085(3-[3-[4-[dideuterio(methylamino)methyl]phenyl]isox...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant FLAG-tagged full length ATR expressed in mammalian cell line co-expressing human recombinant cMyc-tagged full length ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918G5PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381509(CHEMBL2017740)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381517(CHEMBL2017748)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381485(CHEMBL2017593)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240227(CHEMBL4084391)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human His-tagged CSF1R cytoplasmic domain (538 to 910 residues) expressed in baculovirus expression system using fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381509(CHEMBL2017740)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381518(CHEMBL2017751)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381529(CHEMBL2017760)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240210(CHEMBL4084299)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against HSV-1 Ribonucleoside diphosphate reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240209(CHEMBL4068526)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human c-Kit using poly[Glu:Tyr] (4:1) as substrate measured after 2 hrs in presence of [33gammaP]ATP by P18 ion exchange chromatographi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240228(CHEMBL4060882)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate incubated for 2 hrs in presence of [33gammaP]ATP by P81 ion exchange chromatographic...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381515(CHEMBL2017746)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381508(CHEMBL2017618)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381520(CHEMBL2017753)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of [125-I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381520(CHEMBL2017753)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Integral BioSciences, Pvt. Ltd.

Curated by ChEMBL
LigandPNGBDBM50456368(CHEMBL4216036)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918G5PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381506(CHEMBL2017616)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Integral BioSciences Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50240227(CHEMBL4084391)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human His-tagged CSF1R cytoplasmic domain (538 to 910 residues) expressed in baculovirus expression system using fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6GC2PubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381498(CHEMBL2017606)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM35909(2-Hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-ph...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at androgen receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luciferas...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd

Curated by ChEMBL
LigandPNGBDBM50381507(CHEMBL2017617)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human recombinant MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH-induced IP3 accumulation response preincubated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z7485PubMed
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