Compile Data Set for Download or QSAR
Found 32 with Last Name = 'boyd' and Initial = 'mr'
TargetProtein kinase C zeta type(Rattus norvegicus)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478518(CHEMBL514017)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]PDBu from rat brain membrane PKCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8BF5PubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090045((2,3-Dihydroxy-4-methoxy-phenyl)-(3,4,5-trimethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6CFQPubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090044((Z)-2',3'-dihydroxy-3,4,4',5-tetramethoxystilbene ...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6CFQPubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N300QZPubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50006677(1,2,3-Trimethoxy-5-[(Z)-2-(4-methoxy-phenyl)-vinyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N300QZPubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Tested for 50 % inhibition of tubulin polymerization by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064891(5,7,3'-trihydroxy-3,6-4'-trimethoxyflavone | 5,7-D...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for 50 % inhibition of tubulin polymerization by turbidimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5N91
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478521(CHEMBL465805)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50471653(CHEMBL297299)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N300QZPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50292441(1beta-hydroxyaleuritolic acid 3-p-hydroxybenzoate ...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478525(CHEMBL465804)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478526(CHEMBL448121)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478416(CHEBI:65536 | CHEMBL444821)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8J9JPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478527(Aleuritolic Acid 3-P-Hydroxybenzoate | CHEMBL45689...)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478523(Aleuritolic Acid 3-P-Hydroxycinnamate | CHEMBL5033...)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478415(Buchapine | CHEBI:65535)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8J9JPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478524(CHEMBL450856)copy SMILEScopy InChI
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478522(CHEMBL454238)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50471654(CHEMBL44574)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N300QZPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478522(CHEMBL454238)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50090046(CHEMBL329267 | Phosphoric acid mono-[3-methoxy-2-p...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6CFQPubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064259(CHEMBL289351 | Combretastatin A4 phosphate | Di-So...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6CFQPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478528(CHEMBL451536)copy SMILEScopy InChI
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by UIC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478526(CHEMBL448121)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478523(Aleuritolic Acid 3-P-Hydroxycinnamate | CHEMBL5033...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50064259(CHEMBL289351 | Combretastatin A4 phosphate | Di-So...)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+4nMAssay Description:The compound was tested for the concentration to inhibit 50% of tubulin polymerization.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N300QZPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478521(CHEMBL465805)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50292441(1beta-hydroxyaleuritolic acid 3-p-hydroxybenzoate ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478528(CHEMBL451536)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478524(CHEMBL450856)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50478527(Aleuritolic Acid 3-P-Hydroxybenzoate | CHEMBL45689...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase by NCI assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SP1PubMed