Compile Data Set for Download or QSAR
Found 246 with Last Name = 'jain' and Initial = 'mr'
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50178975(4,6-dichloro-5-(4-hydroxy-3-isopropylphenoxy)-1H-i...)copy SMILEScopy InChI
Affinity DataKi:  0.0600nMAssay Description:Binding affinity to TRbeta1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09FJPubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)copy SMILEScopy InChI
Affinity DataKi:  0.370nMAssay Description:Binding affinity to TRbeta1More data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)copy SMILEScopy InChI
Affinity DataKi:  7.18nMAssay Description:Binding affinity to TRalpha1More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMedDrugBank
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  475nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50401076(CHEMBL457748)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Binding affinity to TRbeta1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09FJPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataKi:  1.99E+3nMAssay Description:Displacement of [3H]WIN552122 from human recombinant CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50401076(CHEMBL457748)copy SMILEScopy InChI
Affinity DataKi:  1.25E+4nMAssay Description:Binding affinity to TRalpha1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ09FJPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  2.45E+4nMAssay Description:Displacement of [3H]WIN552122 from human recombinant CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  2.45E+4nMAssay Description:Displacement of [3H]WIN552122 from human recombinant CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50226179((+)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-...)copy SMILEScopy InChI
Affinity DataKi:  2.64E+4nMAssay Description:Displacement of [3H]WIN552122 from human recombinant CB2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81CTKPubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD1 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316499(CHEMBL4167582)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316852(CHEMBL4171446)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316816(CHEMBL4161223)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316816(CHEMBL4161223)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50321025(CHEMBL4170335)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN3(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50446903(CHEMBL3115293)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN3(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317545(CHEMBL4173371)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316844(CHEMBL4162417)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN3(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317465(CHEMBL4165865)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50318459(CHEMBL4159227)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN2(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317547(CHEMBL4163812)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of PHD1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM350280(2-(4-Hydroxy-2-oxo-1-(3'- (trifluoromethoxy)-[1,1'...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50421200(CHEMBL2087289)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in baculovirus infected Sf9 cells after overnight incubation by scinti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70H37PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50421197(CHEMBL2087286)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in baculovirus infected Sf9 cells after overnight incubation by scinti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70H37PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50538416(CHEMBL4644835 | US11236045, Example 25)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WP2PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50318681(CHEMBL4162309)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetProlyl hydroxylase EGLN3(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317547(CHEMBL4163812)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PHD3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317468(CHEMBL4169558)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50538393(CHEMBL4647321 | US11236045, Example 1)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WP2PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50318913(CHEMBL4177137)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of NLRP3 in human THP1 cells assessed as inhibition of IL-1beta productionMore data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50321014(CHEMBL4163550)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50538418(CHEMBL4641961 | US11236045, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WP2PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317078(CHEMBL4170656)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of PHD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM242568(US9422240, 1-378)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of human PHD2 expressed in 293FT cells using HIF-1 [alpha] as substrate after 20 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50538405(CHEMBL4642066)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WP2PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50421198(CHEMBL2087287)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in baculovirus infected Sf9 cells after 16-18 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70H37PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50421198(CHEMBL2087287)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in baculovirus infected Sf9 cells after overnight incubation by scinti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70H37PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50316511(CHEMBL4161082)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of PHD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50320830(CHEMBL4162965)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
Cadila Healthcare Ltd.

Curated by ChEMBL
LigandPNGBDBM50538407(CHEMBL4647621 | US11236045, Example 22)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed human THP1 cells assessed as reduction in IL-1beta level preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WP2PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50320749(CHEMBL4165493)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD2 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
Cadila Healthcare Limited

Curated by ChEMBL
LigandPNGBDBM50317547(CHEMBL4163812)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of PHD2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70JC7PubMed
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