Compile Data Set for Download or QSAR
Found 432 with Last Name = 'cheng' and Initial = 'n'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50381853(CHEMBL2023067)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
LigandPNGBDBM50614520(CHEMBL5271228)copy SMILES
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50381855(CHEMBL2023066)copy SMILEScopy InChI
Affinity DataIC50: 2.34nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50381854(CHEMBL2022467)copy SMILEScopy InChI
Affinity DataIC50: 2.64nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
LigandPNGBDBM50614523(CHEMBL5276678)copy SMILES
Affinity DataIC50: 8.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
LigandPNGBDBM50614533(CHEMBL5267053)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50381856(CHEMBL2022464)copy SMILEScopy InChI
Affinity DataIC50: 13.8nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373415(CHEMBL256713)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of truncated human N-terminal GST-fusion tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using FAM-labelled ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50373415(CHEMBL256713)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of full length human N-terminal GST-fusion tagged IRAK4 expressed in baculovirus expression system using FAM-labelled peptide as substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194448(CHEMBL3972289)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
LigandPNGBDBM50614533(CHEMBL5267053)copy SMILES
Affinity DataIC50: 34nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194466(CHEMBL3958557)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194475(CHEMBL3889586)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194259(CHEMBL3939958)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
LigandPNGBDBM50614521(CHEMBL5272585)copy SMILES
Affinity DataIC50: 45nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50614533(CHEMBL5267053)copy SMILES
Affinity DataIC50: 45nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194476(CHEMBL3942693)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
LigandPNGBDBM50614531(CHEMBL5290950)copy SMILES
Affinity DataIC50: 51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50614522(CHEMBL5273916)copy SMILES
Affinity DataIC50: 51nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50614532(CHEMBL5284612)copy SMILES
Affinity DataIC50: 53nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194477(CHEMBL3916023)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50579721(CHEMBL4798892)copy SMILES
Affinity DataIC50: 60nMAssay Description:Inhibition of truncated human N-terminal GST-fusion tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using FAM-labelled ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194258(CHEMBL3934881)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194448(CHEMBL3972289)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194458(CHEMBL3987134)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50579722(CHEMBL4762381)copy SMILES
Affinity DataIC50: 72nMAssay Description:Inhibition of truncated human N-terminal GST-fusion tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using FAM-labelled ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194466(CHEMBL3958557)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194475(CHEMBL3889586)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194458(CHEMBL3987134)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
LigandPNGBDBM50614524(CHEMBL5286058)copy SMILES
Affinity DataIC50: 75nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194457(CHEMBL3969494)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50579720(CHEMBL5083561)copy SMILES
Affinity DataIC50: 79nMAssay Description:Inhibition of truncated human N-terminal GST-fusion tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using FAM-labelled ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50579719(CHEMBL5075213)copy SMILES
Affinity DataIC50: 80nMAssay Description:Inhibition of truncated human N-terminal GST-fusion tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using FAM-labelled ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3XMHPubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194474(CHEMBL3953637)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194259(CHEMBL3939958)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194447(CHEMBL3978944)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
LigandPNGBDBM50614529(CHEMBL5287682)copy SMILES
Affinity DataIC50: 90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50529830(CHEMBL4540510)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of purified SMS2 (unknown origin) using C6-NBD-Ceramide and DMPC as substrates preincubated for 5 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8C4JPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50529830(CHEMBL4540510)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of purified SMS2 (unknown origin) using C6-NBD-Ceramide and DMPC as substrates preincubated for 5 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8C4JPubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194477(CHEMBL3916023)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Xiangtan University

Curated by ChEMBL
LigandPNGBDBM50437452(CHEMBL2409349)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of bovine lens aldose reductase using DL-glyceraldehyde as substrate assessed as NADPH oxidation measured for 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ67GTPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194258(CHEMBL3934881)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194474(CHEMBL3953637)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194471(CHEMBL3943850)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194466(CHEMBL3958557)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194448(CHEMBL3972289)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194262(CHEMBL3949885)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H1340DPubMed
TargetAldo-keto reductase family 1 member B1 [K65Q](Bos taurus (Cattle))
Xiangtan University

Curated by ChEMBL
LigandPNGBDBM50437469(CHEMBL2409351)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:Inhibition of bovine lens aldose reductase using DL-glyceraldehyde as substrate assessed as NADPH oxidation measured for 10 mins by spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ67GTPubMed
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