Compile Data Set for Download or QSAR
Found 376 with Last Name = 'pala' and Initial = 'n'
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058941(CHEMBL3326411)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232182(CHEMBL4097327)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059068(CHEMBL3326413)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059069(CHEMBL3326414)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50087713((1-Ethyl-propyl)-[3-(4-methoxy-2-methyl-phenyl)-2,...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059070(CHEMBL3326415)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232188(CHEMBL4070141)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058937(CHEMBL3326401)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058941(CHEMBL3326411)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232179(CHEMBL4105538)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232178(CHEMBL4081285)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232182(CHEMBL4097327)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059080(CHEMBL3326409)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059078(CHEMBL3326407)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059076(CHEMBL3326405)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059075(CHEMBL3326404)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232191(CHEMBL4089611)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232188(CHEMBL4070141)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059074(CHEMBL3326403)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232191(CHEMBL4089611)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059072(CHEMBL3326417)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232201(CHEMBL4099753)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058938(CHEMBL3326419)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM15233(4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]benzene...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058937(CHEMBL3326401)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232190(CHEMBL4061482)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059079(CHEMBL3326408)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232201(CHEMBL4099753)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50262063(4-(4-p-tolyl-1H-1,2,3-triazol-1-yl)benzenesulfonam...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058939(CHEMBL3326418)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059070(CHEMBL3326415)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059069(CHEMBL3326414)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232190(CHEMBL4061482)copy SMILEScopy InChI
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059073(CHEMBL3326402)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232183(CHEMBL4097805)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [125I]o-CRF from recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059068(CHEMBL3326413)copy SMILEScopy InChI
Affinity DataKi:  5.30nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059076(CHEMBL3326405)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058940(CHEMBL3326410)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of human CA12 using CO2 as substrate incubated for 6 hrs prior to substrate addition measured for 10 to 100 secs by stopped flow techniqueMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 catalytic domain preincubated for 15 mins prior to testing measured for 10 to 100 secs by pheno...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50262062(4-(4-phenyl-1H-1,2,3-triazol-1-yl)benzenesulfonami...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059075(CHEMBL3326404)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059074(CHEMBL3326403)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232200(CHEMBL4081736)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184RNPubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM15233(4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]benzene...)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50058938(CHEMBL3326419)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University of KwaZulu-Natal

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059078(CHEMBL3326407)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Universit£ di Sassari

Curated by ChEMBL
LigandPNGBDBM50059067(CHEMBL3326412)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated for 15 mins by stopped-flow CO2 hydrase AssayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z68PubMed
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