TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]Pentazocine from rat sigma 1 receptor in rat PC12 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [125I]HEAT from adrenergic alpha2A receptorMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D4 receptorMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]tiotidine from human histamine H2 receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [125I]HEAT from adrenergic Alpha-2C receptorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(MOUSE)
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]citalopram from human SERTMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [125I]HEAT from adrenergic alpha2B receptorMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]alpha-methylhistamine from human histamine H3 receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of [125I]HEAT from adrenergic alpha1A receptorMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 377nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(MOUSE)
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(MOUSE)
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
TargetSodium-dependent noradrenaline transporter(MOUSE)
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(MOUSE)
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2B(Mus musculus (Mouse))
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Mus musculus (Mouse))
National Institutes of Health
Curated by PDSP Ki Database
National Institutes of Health
Curated by PDSP Ki Database
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKd: 7.20nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
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