Compile Data Set for Download or QSAR
Found 106 with Last Name = 'varga' and Initial = 'n'
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359016(CHEMBL1924017)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359013(CHEMBL1924014)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359018(CHEMBL1924019)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359032(CHEMBL1924024)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359022(CHEMBL1924023)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359017(CHEMBL1924018)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359012(CHEMBL1924013)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359023(CHEMBL1170725)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359015(CHEMBL1924016)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359025(CHEMBL1924005)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359024(CHEMBL1924004)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162903(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359014(CHEMBL1924015)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 in hTP binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359024(CHEMBL1924004)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162894(CHEMBL361972 | [2-(4-Fluoro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359021(CHEMBL1924022)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359020(CHEMBL1924021)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162917(CHEMBL360288 | [6-(4-Fluoro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359026(CHEMBL1924006)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162891(CHEMBL179980 | [6-(4-Fluoro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359025(CHEMBL1924005)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359019(CHEMBL1924020)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359033(CHEMBL1924012)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359027(CHEMBL1924007)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359028(CHEMBL1924008)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162896(CHEMBL369330 | [3-tert-Butyl-6-(4-fluoro-benzenesu...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359029(CHEMBL1924009)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162901(CHEMBL180733 | [5-(4-Fluoro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162897(3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162897(3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibitory activity of the compound against CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359026(CHEMBL1924006)copy SMILEScopy InChI
Affinity DataKi:  251nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50161746((R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Inhibitory concentration of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calciumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359031(CHEMBL1924011)copy SMILEScopy InChI
Affinity DataKi:  631nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359030(CHEMBL1924010)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162925(3-[6-(2-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  970nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359028(CHEMBL1924008)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162902(3-(6-Benzenesulfonylamino-1,2,3,4-tetrahydro-carba...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359027(CHEMBL1924007)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359023(CHEMBL1170725)copy SMILEScopy InChI
Affinity DataKi:  1.26E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162892(3-[6-(3-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162897(3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 in hTP binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359030(CHEMBL1924010)copy SMILEScopy InChI
Affinity DataKi:  1.59E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162906(3-[6-(3-Chloro-4-fluoro-benzenesulfonylamino)-1,2,...)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162918(3-[6-(4-Methoxy-benzenesulfonylamino)-1,2,3,4-tetr...)copy SMILEScopy InChI
Affinity DataKi:  2.10E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Athersys, Inc.

Curated by ChEMBL
LigandPNGBDBM50162898(2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetra...)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity of the compound for binding of PGD-2 to CRTH-2 in hCRTH-2 binding assay using HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P0ZHTPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359029(CHEMBL1924009)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50359031(CHEMBL1924011)copy SMILEScopy InChI
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrs in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C6DPubMed
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