Compile Data Set for Download or QSAR
Found 919 with Last Name = 'kallan' and Initial = 'nc'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104202(US8575145, 79)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104204(US8575145, 81)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM41535(US8575145, 106 | US8575145, 66)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104229(US8575145, 106)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104162(US8575145, 39)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104187(US8575145, 64)copy SMILEScopy InChI
Affinity DataIC50: 0.640nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104140(US8575145, 17)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104186(US8575145, 63)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104142(US8575145, 19)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104237(US8575145, 114)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104221(US8575145, 98)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104193(US8575145, 70)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104165(US8575145, 42)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104188(US8575145, 65)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104147(US8575145, 24)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM41535(US8575145, 106 | US8575145, 66)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-3(Rattus norvegicus (Rat))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104213(US8575145, 120 | US8575145, 121 | US8575145, 150 |...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104246(US8575145, 123)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)copy SMILEScopy InChI
Affinity DataIC50: 0.920nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104190(US8575145, 67)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104196(US8575145, 73)copy SMILEScopy InChI
Affinity DataIC50: 0.960nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array BioPharma

Curated by ChEMBL
LigandPNGBDBM50446312(CHEMBL3109350)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N24VQPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104215(US8575145, 152 | US8575145, 92 | US8575145, 92/122)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array BioPharma

Curated by ChEMBL
LigandPNGBDBM50446319(CHEMBL3109343)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N24VQPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc

Curated by ChEMBL
LigandPNGBDBM50327782((R)-2-amino-3-(4-chlorophenyl)-1-(4-(5-methyl-7H-p...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908XQPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc

Curated by ChEMBL
LigandPNGBDBM50327785((R)-2-amino-1-(4-(5-chloro-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908XQPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc

Curated by ChEMBL
LigandPNGBDBM50332316((R)-2-amino-3-(4-chlorophenyl)-1-(4-((S)-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BBJPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc

Curated by ChEMBL
LigandPNGBDBM50332329((S)-2-(4-chlorobenzyl)-3-(isopropylamino)-1-(4-((S...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Akt1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BBJPubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc.

Curated by ChEMBL
LigandPNGBDBM50398382(CHEMBL2177387)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P1160PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104169(US8575145, 46/47/48/49/50 | US8575145, 77 | US8575...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104139(US8575145, 16)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104255(US8575145, 132)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104248(US8575145, 125)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104240(US8575145, 117)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104241(US8575145, 118/119 | US8575145, 149)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104191(US8575145, 68)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104226(US8575145, 103)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104238(US8575145, 115)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104222(US8575145, 130 | US8575145, 99/100)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104141(US8575145, 18)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104256(US8575145, 133)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104124(US8575145, 1)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104192(US8575145, 69)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104233(US8575145, 110)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Array BioPharma Inc.

Curated by ChEMBL
LigandPNGBDBM50398358(CHEMBL2177361)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P1160PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Array BioPharma Inc.

US Patent
LigandPNGBDBM104208(US8575145, 85)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled pe...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M90797US Patent
TargetPlatelet-derived growth factor receptor beta(Mus musculus (mouse))
Array BioPharma

Curated by ChEMBL
LigandPNGBDBM50446315(CHEMBL3109347)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PDGF-induced PDGFRbeta phosphorylation in mouse NIH3T3 cells incubated for 1 hr prior to PDGF induction measured after 15 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N24VQPubMed
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