Compile Data Set for Download or QSAR
Found 278 with Last Name = 'shaikh' and Initial = 'ns'
LigandPNGBDBM555248(USRE49080, Example 16)copy SMILES
Affinity DataIC50: 0.150nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555247(USRE49080, Example 15)copy SMILES
Affinity DataIC50: 0.200nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555251(USRE49080, Example 21)copy SMILES
Affinity DataIC50: 0.200nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555242(USRE49080, Example 8)copy SMILES
Affinity DataIC50: 0.25nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555255(USRE49080, Example 28)copy SMILES
Affinity DataIC50: 0.330nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555263(USRE49080, Example 42)copy SMILES
Affinity DataIC50: 0.350nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555252(USRE49080, Example 22)copy SMILES
Affinity DataIC50: 0.400nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM50560402(LIK-066 | Licogliflozin | Lik066 | USRE49080, Exam...)copy SMILES
Affinity DataIC50: 0.5nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555250(USRE49080, Example 20)copy SMILES
Affinity DataIC50: 0.550nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555249(USRE49080, Example 17)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555270(USRE49080, Example 66)copy SMILES
Affinity DataIC50: 0.900nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM364370(4-[3-(2,6-dichlorobenzoyl)-7-fluoro-1H-indol-1-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512498(CHEMBL4570491)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555271(USRE49080, Example 69)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555257(USRE49080, Example 31)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555253(USRE49080, Example 24)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555245(USRE49080, Example 11)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555254(USRE49080, Example 25)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555272(USRE49080, Example 71)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512490(CHEMBL4454027)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512497(CHEMBL4567440)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50203542(CHEMBL3218921)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555267(USRE49080, Example 60)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555269(USRE49080, Example 65)copy SMILES
Affinity DataIC50: 2.70nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555238(USRE49080, Example 1)copy SMILES
Affinity DataIC50: 2.70nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512504(CHEMBL4540580)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555264(USRE49080, Example 43)copy SMILES
Affinity DataIC50: 3.90nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM364371(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-1 H-ind...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512525(CHEMBL4454020)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555246(USRE49080, Example 14)copy SMILES
Affinity DataIC50: 5.5nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393129(CHEMBL2153461)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DG6PubMed
TargetSuccinate receptor 1(Rat)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DG6PubMed
LigandPNGBDBM555243(USRE49080, Example 9)copy SMILES
Affinity DataIC50: 7.20nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512506(CHEMBL4551954)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Inverse agonist activity at GST-tagged RORgammat LBD (unknown origin) using fluorescein-D22 co-activator peptide as substrate incubated for 1 hr by T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555267(USRE49080, Example 60)copy SMILES
Affinity DataIC50: 9nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555259(USRE49080, Example 35)copy SMILES
Affinity DataIC50: 9.5nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512497(CHEMBL4567440)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512510(CHEMBL4561072)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
LigandPNGBDBM555258(USRE49080, Example 33)copy SMILES
Affinity DataIC50: 11nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM364371(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-1 H-ind...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512495(CHEMBL4466120)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393123(CHEMBL2153446)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DG6PubMed
LigandPNGBDBM555239(USRE49080, Example 2)copy SMILES
Affinity DataIC50: 11.1nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM364370(4-[3-(2,6-dichlorobenzoyl)-7-fluoro-1H-indol-1-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393133(CHEMBL2153465)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DG6PubMed
LigandPNGBDBM555265(USRE49080, Example 46)copy SMILES
Affinity DataIC50: 14nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
LigandPNGBDBM555261(USRE49080, Example 38)copy SMILES
Affinity DataIC50: 14.4nMAssay Description:The SGLT-2 assay is carried out as follows: CHO-hSGLT2 cells are cultivated in Ham's F12 Medium (BioWhittaker) with 10% foetal calf serum and 250...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868J4US Patent
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512491(CHEMBL4556521)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
TargetSuccinate receptor 1(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393122(CHEMBL2153445)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DG6PubMed
TargetNuclear receptor ROR-gamma(Human)
Advinus Therapeutics Limited

Curated by ChEMBL
LigandPNGBDBM50512502(CHEMBL4577409)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Transactivation of recombinant GAL4-DBD fused RORgammat LBD (unknown origin) expressed in HEK293T cells incubated for 18 to 24 hrs by dual-Glo lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50R96PubMed
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