TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rattus norvegicus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of Wistar rat heart SERCA2a after 1 hrMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(RAT)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of Wistar rat kidney Na+,K+-ATPase alpha1 after 2 hrsMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rattus norvegicus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Wistar rat EDL muscle SERCA1a after 1 hrMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 7.50E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 9.65E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 1.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 3.21E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 4.81E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 2.23E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 2.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 2.70E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 5.00E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 3.15E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 0.200nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg
Curated by ChEMBL
Albert Ludwigs University Freiburg
Curated by ChEMBL
Affinity DataKd: 1.03E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair