Compile Data Set for Download or QSAR
Found 17 with Last Name = 'fedosova' and Initial = 'nu'
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rattus norvegicus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)copy SMILEScopy InChI
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of Wistar rat heart SERCA2a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(RAT)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)copy SMILEScopy InChI
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of Wistar rat kidney Na+,K+-ATPase alpha1 after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rattus norvegicus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)copy SMILEScopy InChI
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Wistar rat EDL muscle SERCA1a after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097547(CHEMBL3125413)copy SMILEScopy InChI
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097548(CHEMBL3586098)copy SMILEScopy InChI
Affinity DataKd:  9.65E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097555(CHEMBL3586095)copy SMILEScopy InChI
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097550(CHEMBL3125412)copy SMILEScopy InChI
Affinity DataKd:  3.21E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097551(CHEMBL3125420)copy SMILEScopy InChI
Affinity DataKd:  4.81E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097552(CHEMBL3125415)copy SMILEScopy InChI
Affinity DataKd:  2.23E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097553(CHEMBL3586096)copy SMILEScopy InChI
Affinity DataKd:  2.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097554(Casearborin D)copy SMILEScopy InChI
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097556(Alisol B | CHEBI:81104)copy SMILEScopy InChI
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097557(CHEMBL3586100)copy SMILEScopy InChI
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097535(CHEMBL3125414)copy SMILEScopy InChI
Affinity DataKd:  3.15E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097525(CHEMBL3586099)copy SMILEScopy InChI
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(CHEMBL96926 | OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4...)copy SMILEScopy InChI
Affinity DataKd:  0.200nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Oryctolagus cuniculus)
Albert Ludwigs University Freiburg

Curated by ChEMBL
LigandPNGBDBM50097549(CHEMBL3586097)copy SMILEScopy InChI
Affinity DataKd:  1.03E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TR2PubMed