Compile Data Set for Download or QSAR
Found 311 with Last Name = 'monteiro' and Initial = 'o'
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505576(CHEMBL4458252)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of G9a (unknown origin) by scintillation proximity AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0JPZPubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505574(CHEMBL4451634)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0JPZPubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505583(CHEMBL4573889)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505578(CHEMBL4570122)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0JPZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505582(CHEMBL4465568)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of G9a (unknown origin) by scintillation proximity AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetBromodomain-containing protein 1(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 128nMAssay Description:Alphascreen assay. Binding to BRD1A (domain start/stop: E556-A688) by alphascreen assayMore data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2A(Homo sapiens (Human))
Cancer Research UK Cancer Therapeutics Unit

Curated by ChEMBL
LigandPNGBDBM50078630(CHEMBL4296718)copy SMILEScopy InChI
Affinity DataIC50: 136nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505573(CHEMBL4577068)copy SMILEScopy InChI
Affinity DataIC50: 152nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
Cancer Research UK Cancer Therapeutics Unit

Curated by ChEMBL
LigandPNGBDBM50078630(CHEMBL4296718)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862M28PubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:Binding affinity to recombinant human His-tagged SPIN1 (49 to 262 residues) expressed in Escherichia coli BL21 (DE3) incubated for 30 mins by AlphaLI...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50078631(CHEMBL4650212)copy SMILEScopy InChI
Affinity DataIC50: 189nMAssay Description:Homogeneous Time Resolved Fluorescence (HTRF) assay. Domain start/stop: L14-Q143More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T0JPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetTranscription activator BRG1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50266286(CHEMBL4650213)copy SMILEScopy InChI
Affinity DataIC50: 263nMAssay Description:Alphascreen assay. Binding to SMARCA4A (domain start/stop: L1451-E1580) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75KX6PubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148463(CHEMBL3770971)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148467(CHEMBL3770004)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 282nMAssay Description:Alphascreen assay. Binding to BRPF1B (domain start/stop: M626-G740) by alphascreen assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148468(CHEMBL3769887)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148465(CHEMBL3771151)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148464(CHEMBL3771106)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 311nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50266292(CHEMBL3906203)copy SMILEScopy InChI
Affinity DataIC50: 324nMAssay Description:Alphascreen assay. Binding to CREBBPA (domain start/stop: R1081-G1197) by alphascreen assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148460(CHEMBL1346130)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148478(CHEMBL3769965 | US10702504, Compound A)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505579(CHEMBL4591023)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148470(CHEMBL3771002)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505571(CHEMBL4528213)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7S2SPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148549(4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 383nMAssay Description:Alphascreen assay. Binding to BRPF1B (domain start/stop: M626-G740) by alphascreen assayMore data for this Ligand-Target Pair
TargetSpindlin-1(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50505570(CHEMBL4476309)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Displacement of trimethylated biotinylated histone H3 peptide from recombinant human His-tagged SPIN1 (26 to 262 residues) expressed in Escherichia c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTranscription activator BRG1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50266286(CHEMBL4650213)copy SMILEScopy InChI
Affinity DataIC50: 411nMAssay Description:Alphascreen assay. Binding to SMARCA4A (domain start/stop: L1451-E1580) by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75KX6PubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148462(CHEMBL3770886)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148478(CHEMBL3769965 | US10702504, Compound A)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of N-terminal His6-SUMO-1-tagged recombinant human TRIM24 bromodomain expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells by Alpha Scr...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148475(CHEMBL3770465)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetPeregrin(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148476(CHEMBL3770391)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)copy SMILEScopy InChI
Affinity DataIC50: 468nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148468(CHEMBL3769887)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of N-terminal His6-SUMO-1-tagged recombinant human TRIM24 bromodomain expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells by Alpha Scr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9S9GPubMed
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