Compile Data Set for Download or QSAR
Found 231 with Last Name = 'ryabtsova' and Initial = 'o'
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382287(CHEMBL2024671)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli assessed as pNA release from Z-Gly-Pro-p-nitroanilide pre-incubated with enzyme fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434165(CHEMBL2385271 | US9346814, Cmpd No 11 Example 14)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434170(CHEMBL2385299 | US9346814, Cmpd No 21 Example 25)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human seminal plasma DPP4 assessed as pNA release from Gly-Pro-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human seminal plasma DPP4 assessed as pNA release from Gly-Pro-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...More data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of human seminal plasma DPP2 assessed as pNA release from Lys-Ala-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434191(CHEMBL2385278)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382283(CHEMBL2022530 | US9346814, Ref. Cmpd No 1 (Example...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of human seminal plasma DPP4 assessed as pNA release from Gly-Pro-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMedDrugBank
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382281(CHEMBL2022528)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434190(CHEMBL2385279)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434171(CHEMBL2385298 | US9346814, Cmpd No 38 Example 43)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434174(CHEMBL2385295)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382262(CHEMBL2022507)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli assessed as pNA release from Z-Gly-Pro-p-nitroanilide pre-incubated with enzyme fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434183(CHEMBL2385286)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434160(CHEMBL2385276)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50326374((S)-N-(2-(2-cyanopyrrolidin-1-yl)-2-oxoethyl)-1-na...)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434172(CHEMBL2385297)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382282(CHEMBL2022529)copy SMILEScopy InChI
Affinity DataIC50: 850nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 860nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli assessed as pNA release from Z-Gly-Pro-p-nitroanilide pre-incubated with enzyme fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434174(CHEMBL2385295)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434173(CHEMBL2385296)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382281(CHEMBL2022528)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli assessed as pNA release from Z-Gly-Pro-p-nitroanilide pre-incubated with enzyme fo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50382274(CHEMBL2022521)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2W5PPubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
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