Compile Data Set for Download or QSAR
Found 296 with Last Name = 'cotelle' and Initial = 'p'
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50021581(CHEMBL414850 | L-870810)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50021581(CHEMBL414850 | L-870810)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of HIV1 integrase using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39K5PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50021581(CHEMBL414850 | L-870810)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50021581(CHEMBL414850 | L-870810)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of HIV1 integrase strand transfer activity using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39K5PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of strand transfer activity of HIV1 integrase using pre-cleaved oligonucleotide as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017364(CHEMBL3288273)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017362(CHEMBL3288268)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017359(CHEMBL3288265)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017358(CHEMBL3286416)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492499(CHEMBL2407278)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMedDrugBank
TargetCytochrome P450 2D6(Homo sapiens (Human))
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50410855(CIN-QUIN | QUINIDEX | QUINIDINE SULFATE)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant CYP2D6 (unknown origin) using 7-methoxy-4-trifluoromethylcoumarin as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CYP2D6 using MFC as substrate incubated for 40 mins by fluorimetryMore data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50479372(CHEMBL456326)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017350(CHEMBL3288281)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492504(CHEMBL2407277)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells assessed as inhibition of tail current after 5 mins by automated whole-cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2J1PPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of human ERG tail current by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50271260(CHEMBL4130196)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human His-tagged YAP (50 to 171 residues) interaction with human GST-tagged TEAD1 (194 to 411) expressed in Escherichia coli BL21(DE3) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91H7PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of HIV1 integrase using labelled U5A/U5B double stranded DNA substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39K5PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017365(CHEMBL3288274)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017360(CHEMBL3288266)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50237838((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(4,5-dihy...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV1 integrase using labelled U5A/U5B double stranded DNA substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39K5PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492515(CHEMBL2407272)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492507(CHEMBL2407280)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of strand transfer activity of HIV1 integrase using pre-cleaved oligonucleotide as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492502(CHEMBL2407284)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492505(CHEMBL2407283)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492508(CHEMBL2407287)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017356(CHEMBL3288263)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017357(CHEMBL3288264)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017349(CHEMBL3288280)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492508(CHEMBL2407287)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of 3'-processing activity of HIV1 integrase using 32P-5'-TGTGGAAAATCTCTAGCAGT-3' and 5'-ACTGCTAGAGATTTTCCACA-3' as substrate after 1 hr by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017361(CHEMBL3288267)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50237838((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(4,5-dihy...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of HIV1 integrase strand transfer activity using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M39K5PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017351(CHEMBL3288282)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492503(CHEMBL2407281)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492507(CHEMBL2407280)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV1 integrase overall inhibition using 5'-digoxigenin-labeled 5'-GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ Lille Nord de France

Curated by ChEMBL
LigandPNGBDBM50017353(CHEMBL3288271)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of HIV-1 overall integrase activity using 5'-digoxigenin-labeled GACCCTTTTAGTCAGTGTGGAAAATCTCTAGCAGT-3' as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ6335PubMed
TargetTranscriptional enhancer factor TEF-1(Homo sapiens)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50271259(CHEMBL4129172)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of Gal4-fused TEAD 1 (unknown origin) interaction with YAP expressed in human 293T cells by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91H7PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492503(CHEMBL2407281)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of strand transfer activity of HIV1 integrase using pre-cleaved oligonucleotide as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50170903(CHEMBL3805993)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of HIV1 integrase using 3'-biotin-labelled and 5'-digoxigenin-labelled oligonucleotide substrate incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2J1PPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50170903(CHEMBL3805993)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of HIV1 integrase using 3'-biotin-labelled and 5'-digoxigenin-labelled oligonucleotide substrate incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2J1PPubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50479373(CHEMBL512021)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XJ1PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£ de Lille 1

Curated by ChEMBL
LigandPNGBDBM50492508(CHEMBL2407287)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Inhibition of strand transfer activity of HIV1 integrase using pre-cleaved oligonucleotide as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ06QTPubMed
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