Compile Data Set for Download or QSAR
Found 57 with Last Name = 'dubreuil' and Initial = 'p'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024328(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GRTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)copy SMILEScopy InChI
Affinity DataIC50: 152nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)copy SMILEScopy InChI
Affinity DataIC50: 171nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)copy SMILEScopy InChI
Affinity DataIC50: 206nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)copy SMILEScopy InChI
Affinity DataIC50: 228nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024330(3-(3-Benzyl-ureido)-3-{2-[2-tert-butoxycarbonylami...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GRTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)copy SMILEScopy InChI
Affinity DataIC50: 321nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359983(CHEMBL1927769)copy SMILEScopy InChI
Affinity DataIC50: 559nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)copy SMILEScopy InChI
Affinity DataIC50: 607nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359985(CHEMBL1927772)copy SMILEScopy InChI
Affinity DataIC50: 760nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359986(CHEMBL1927625)copy SMILEScopy InChI
Affinity DataIC50: 793nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)copy SMILEScopy InChI
Affinity DataIC50: 811nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024327(CHEMBL349888 | N-{1-[2-tert-Butoxycarbonylamino-3-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GRTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TPR-fused MET-mediated mouse BA/F3 cell proliferation after 48 hrs by cell titre blue based spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359985(CHEMBL1927772)copy SMILEScopy InChI
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024332(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibitory activity for binding of [125I]-(Nle11)-HG-13 to gastrin receptor on isolated rabbit gastric mucosal cells.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4GRTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359987(CHEMBL1927778)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
CNRS UMR 6216

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)copy SMILEScopy InChI
Affinity DataIC50: 7.73E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8FZTPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
Displayed 1 to 50 (of 57 total ) | Next | Last >>
Jump to: