Compile Data Set for Download or QSAR
Found 104 with Last Name = 'grant' and Initial = 'p'
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517230(CHEMBL4467984)copy SMILEScopy InChI
Affinity DataKi:  0.840nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517232(CHEMBL4546839)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517229(CHEMBL4541515)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517236(CHEMBL4465127)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517222(CHEMBL4579585)copy SMILEScopy InChI
Affinity DataKi:  4.20nMAssay Description:Binding affinity to human D2RMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517233(CHEMBL4568756)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517221(CHEMBL4554135)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50010289((R)6-(Phenethyl-propyl-amino)-5,6,7,8-tetrahydro-n...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H] spiperone from human D2 dopamine receptor expressed in monkey caudate-putamen membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517223(CHEMBL4471116)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517226(CHEMBL4449666)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517227(CHEMBL4562705)copy SMILEScopy InChI
Affinity DataKi:  97nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517225(CHEMBL4453578)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517224(CHEMBL4443273)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517234(CHEMBL4446228)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517235(CHEMBL4444520)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517231(CHEMBL4517197)copy SMILEScopy InChI
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50517228(CHEMBL4461338)copy SMILEScopy InChI
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1R in HEK293 cell membranes after 60 mins liquid scintillation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QW7PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human CAMK1A using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1G(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human CAMK1G using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human CAMK1A using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1B(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human CAMK1B using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083722(CHEMBL3423198)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083725(CHEMBL3423195)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50249319(2-(2-aminoethylamino)-4-(3-(trifluoromethyl)phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human SYK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083722(CHEMBL3423198)copy SMILEScopy InChI
Affinity DataIC50: 9.60nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1B(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human CAMK1B using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545587(CHEMBL4633229 | US11530193, Example 135)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545587(CHEMBL4633229 | US11530193, Example 135)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545573(CHEMBL4635883 | US11530193, Example 54)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human MEK5 using ERK5 as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human CAMK1D using KKALRRQETVDAL as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545586(CHEMBL4632457 | US11530193, Example 106)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545586(CHEMBL4632457 | US11530193, Example 106)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of HA-tagged CAMK1D (unknown origin) expressed in human MDA-MB-231 cells assessed as reduction in CAMK1D autophosphorylation measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545576(CHEMBL4640712 | US11530193, Example 50)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083728(CHEMBL3423193)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetCalcium/calmodulin-dependent protein kinase type 1D(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50545583(CHEMBL4644948)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human full-length His-tagged CAMK1D expressed in baculovirus expression system using autocamtide-2 as substrate preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083718(CHEMBL3423202)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083726(CHEMBL3423194)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083726(CHEMBL3423194)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083725(CHEMBL3423195)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human MLK3 using myelin basic protein as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of human PIM1 using KKRNRTLTK as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083728(CHEMBL3423193)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human BLK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083723(CHEMBL3423197)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of transglutaminase 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50083718(CHEMBL3423202)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q261121GPubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50419254(CHEMBL1835063)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of human SYK using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XG3PubMed
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