Compile Data Set for Download or QSAR
Found 847 with Last Name = 'grieco' and Initial = 'p'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)copy SMILES
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DS4PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134955(CHEMBL2370968 | H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Binding affinity against human Melanocortin 3 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134955(CHEMBL2370968 | H-Tyr-Val-Nle-Gly-Pro-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Binding affinity against Melanocortin 4 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DS4PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413764(CHEMBL504097)copy SMILEScopy InChI
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)copy SMILES
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)copy SMILES
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)copy SMILES
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413762(CHEMBL509604)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DS4PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  0.810nMAssay Description:Binding affinity against human Melanocortin 3 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)copy SMILEScopy InChI
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114077(6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114085((O)C-(C6H4)-C(O)-c[His-D-Phe-Arg-Trp-Lys]-NH2) (MK...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114083(9-Benzyl-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114077(6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114083(9-Benzyl-12-(3H-imidazol-4-ylmethyl)-3-(1H-indol-3...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114088(9-Benzyl-6-(3-guanidino-propyl)-3-(1H-indol-3-ylme...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human melanocortin 5 receptor (hMC5R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114077(6-(3-Guanidino-propyl)-12-(3H-imidazol-4-ylmethyl)...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity against human Melanocortin 5 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114079(15-(2-Acetylamino-hexanoylamino)-9-benzyl-6-(3-gua...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity for human Melanocortin-4 receptor (hMC4R)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)copy SMILES
Affinity DataKi:  1nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)copy SMILES
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114079(15-(2-Acetylamino-hexanoylamino)-9-benzyl-6-(3-gua...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Binding affinity for human Melanocortin-3 receptor (hMC3R) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RB75B3PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50473964(CHEMBL2370836)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FR00C5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50473964(CHEMBL2370836)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DS4PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134947(CHEMBL2370963 | H-Tyr-Val-Nle-Gly-His-Phe-Arg-D-Na...)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity against Melanocortin 4 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413763(CHEMBL448403)copy SMILEScopy InChI
Affinity DataKi:  1.66nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50517327(CHEMBL4472928)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6PRVPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50517320(CHEMBL4568153)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6PRVPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)copy SMILES
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)copy SMILES
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)copy SMILES
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)copy SMILES
Affinity DataKi:  2nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50048702(CHEMBL3315149)copy SMILES
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50517312(CHEMBL4526244)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6PRVPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134954(CHEMBL439128 | H-Tyr-Val-Nle-c[Cys-His-Phe-Arg-Trp...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding affinity against Melanocortin 4 receptor by gamma-MCH displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SJ1K0PPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50413777(CHEMBL524855)copy SMILEScopy InChI
Affinity DataKi:  2.63nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6DFTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50517325(CHEMBL4590360)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6PRVPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50131874(Ac-c[Cys-Glu-His-D-Nal(2')-Arg-Trp-Gly-Cys]-Pro-Pr...)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Inhibitory activity against human melanocortin receptor human Melanocortin 4 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125TDTPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50517316(CHEMBL4462940)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6PRVPubMed
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