Compile Data Set for Download or QSAR
Found 47 with Last Name = 'kapadnis' and Initial = 'p'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362181(({7-[2-(1H-1,2,3-benzotriazol-1-yl)-2-({6-bromo-7-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362195(CHEMBL1938828)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362196(CHEMBL1938829)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362191(CHEMBL1938824)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362192(CHEMBL1938825)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362186(CHEMBL1938819)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362197(CHEMBL1938830)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362183(CHEMBL1938816)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362198(CHEMBL1938831)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362193(CHEMBL1938826)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362194(CHEMBL1938827)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362185(CHEMBL1938818)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50171096(CHEMBL371929 | {4-[[3-Bromo-4-(difluoro-phosphono-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362184(CHEMBL1938817)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362182(CHEMBL1938815)copy SMILEScopy InChI
Affinity DataIC50: 288nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362190(CHEMBL1938823)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362188(CHEMBL1938821)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362189(CHEMBL1938822)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362187(CHEMBL1938820)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of PTP1B assessed as para-nitrophenyl phosphate catalyzed hydrolysis of para-nitrophenol by p-NPP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362181(({7-[2-(1H-1,2,3-benzotriazol-1-yl)-2-({6-bromo-7-...)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362186(CHEMBL1938819)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50171096(CHEMBL371929 | {4-[[3-Bromo-4-(difluoro-phosphono-...)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362195(CHEMBL1938828)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362183(CHEMBL1938816)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
M.S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50362196(CHEMBL1938829)copy SMILEScopy InChI
Affinity DataIC50: 990nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2X05PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259048(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  7.43E+3nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259093(1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)...)copy SMILEScopy InChI
Affinity DataEC50:  7.55E+3nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253755(5-(5-Chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  580nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253755(5-(5-Chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  2.37E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253704(5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  400nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253704(5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  2.32E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259006(1-(2,4-dichlorophenyl)-5-(5-iodothiophen-2-yl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  320nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259006(1-(2,4-dichlorophenyl)-5-(5-iodothiophen-2-yl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  2.94E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259091(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  540nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259091(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  2.59E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259092(5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  1.95E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259092(5-(5-bromothiophen-2-yl)-1-(2,4-dichlorophenyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  510nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataEC50:  240nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMedDrugBank
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)copy SMILEScopy InChI
Affinity DataEC50:  3.12E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259047(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259047(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  2.09E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253756(CHEMBL461862 | N-(Azepan-1-yl)-5-(5-chlorothiophen...)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50253756(CHEMBL461862 | N-(Azepan-1-yl)-5-(5-chlorothiophen...)copy SMILEScopy InChI
Affinity DataEC50:  1.28E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259048(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-4...)copy SMILEScopy InChI
Affinity DataEC50:  690nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259049(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-N...)copy SMILEScopy InChI
Affinity DataEC50:  800nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259049(5-(5-chlorothiophen-2-yl)-1-(2,4-dichlorophenyl)-N...)copy SMILEScopy InChI
Affinity DataEC50:  1.57E+4nMAssay Description:Antagonist activity at human cannabinoid CB2 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50259093(1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)...)copy SMILEScopy InChI
Affinity DataEC50:  1.33E+3nMAssay Description:Antagonist activity at human cannabinoid CB1 receptor expressed in CHOK1 cells assessed as cAMP activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16SPPubMed