Compile Data Set for Download or QSAR
Found 72 with Last Name = 'laduron' and Initial = 'p'
TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataKi:  0.170nMAssay Description:Evaluated for binding activity against [3H]ketanserin as radioligand for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetHistamine H1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Compound was evaluated for binding activity against [3H]-WB- 4101 as radioligand for alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataKi:  164nMAssay Description:Compound was evaluated for binding activity against [3H]-haloperidol as radioligand for Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataKi:  4.42E+3nMAssay Description:Compound was evaluated for binding activity against [3H]haloperidol as radioligand for Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047103(2-{3-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047108(2-{2-[4-(6-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047089(2-{3-[4-(5-Fluoro-1H-indol-3-yl)-3,6-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047092(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047100(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataIC50: 0.562nMAssay Description:Evaluated for binding activity against [3H]ketanserin as radioligand for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047097(2-{2-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047086(2-{3-[4-(1-Methyl-1H-indol-3-yl)-3,6-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047110(2-{4-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047091(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-3,6-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047098(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047106(2-{3-[4-(5-Chloro-1H-indol-3-yl)-3,6-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047105(2-(2-{4-[2-(5-Fluoro-1H-indol-3-yl)-ethyl]-piperid...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047102(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047109(2-{3-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetHistamine H1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047107(2-{2-[4-(5-Fluoro-1H-indol-2-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047095(2-{3-[4-(1H-Indol-3-yl)-piperidin-1-yl]-propyl}-2H...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047085(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperazin-1...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047088(2-{2-[4-(3H-Inden-1-ylmethyl)-piperidin-1-yl]-ethy...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047094(2-{2-[4-(4-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047096(2-{3-[4-(5-Bromo-1H-indol-3-yl)-3,6-dihydro-2H-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047087(1-(3-{1-[3-(1,1-Dioxo-1H-1lambda*6*-naphtho[1,8-cd...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047099(2-{3-[4-(5-Methoxy-1H-indol-3-yl)-3,6-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047090(3-{1-[3-(1,1-Dioxo-1H-1lambda*6*-naphtho[1,8-cd]is...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047095(2-{3-[4-(1H-Indol-3-yl)-piperidin-1-yl]-propyl}-2H...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047089(2-{3-[4-(5-Fluoro-1H-indol-3-yl)-3,6-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for binding activity against [3H]pyrilamine as radioligand for Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9B3NPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047093(CHEMBL19228 | Naphthalene-2-sulfonic acid {2-[4-(5...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047096(2-{3-[4-(5-Bromo-1H-indol-3-yl)-3,6-dihydro-2H-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047093(CHEMBL19228 | Naphthalene-2-sulfonic acid {2-[4-(5...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047106(2-{3-[4-(5-Chloro-1H-indol-3-yl)-3,6-dihydro-2H-py...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047090(3-{1-[3-(1,1-Dioxo-1H-1lambda*6*-naphtho[1,8-cd]is...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047103(2-{3-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047108(2-{2-[4-(6-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Centre de Recherches de Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50047084(10-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of [3H]-peroxitine binding to rat cortical membranes as measure of inhibitory activity towards 5-HT uptakeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047092(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047097(2-{2-[4-(1H-Indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047094(2-{2-[4-(4-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047098(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029154(5-Fluoro-3-piperidin-4-ylmethyl-1H-indole | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047099(2-{3-[4-(5-Methoxy-1H-indol-3-yl)-3,6-dihydro-2H-p...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50047087(1-(3-{1-[3-(1,1-Dioxo-1H-1lambda*6*-naphtho[1,8-cd...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity at dopamine receptor D2 by the inhibition of binding to [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MC8Z3ZPubMed
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