Compile Data Set for Download or QSAR
Found 109 with Last Name = 'lapointe' and Initial = 'p'
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444488(CHEMBL3092613)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444487(CHEMBL3092631)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444486(CHEMBL3091475)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444485(CHEMBL3092620)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444484(CHEMBL3092629)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444483(CHEMBL3092614)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444482(CHEMBL3092628)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444481(CHEMBL3092633)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444480(CHEMBL3092632)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444479(CHEMBL3092619)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444478(CHEMBL3092625)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444477(CHEMBL3092621)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444476(CHEMBL3092617)copy SMILEScopy InChI
Affinity DataKi:  560nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444475(CHEMBL3092615)copy SMILEScopy InChI
Affinity DataKi:  620nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444474(CHEMBL3092624)copy SMILEScopy InChI
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444473(CHEMBL3092622)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444472(CHEMBL3092623)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444471(CHEMBL3092616)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444470(CHEMBL3092626)copy SMILEScopy InChI
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444469(CHEMBL3092618)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444468(CHEMBL3092627)copy SMILEScopy InChI
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50444467(CHEMBL3092630)copy SMILEScopy InChI
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [beta-33P]-2MeS-ADP from human P2Y1 receptor transfected in HEK293 cells after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ630TPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176023(US10047103, 56 | US9688695, 56)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176082(US10047103, 115 | US9688695, 115)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176053(US10047103, 86 | US9688695, 86)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175970(US10047103, 3 | US9605024, Example 3 | US9688695, ...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176039(US10047103, 72 | US9688695, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600788(CHEMBL5206065)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176007(US10047103, 40 | US9688695, 40)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176003(US10047103, 36 | US9688695, 36)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176061(US10047103, 94 | US9688695, 94)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600792(CHEMBL5189522)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175988(US10047103, 21 | US9688695, 21)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286418(US9518064, Example 34)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286424(US9518064, Example 40)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286419(US9518064, Example 35)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176019(US10047103, 52 | US9688695, 52)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176026(US10047103, 59 | US9688695, 59)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176258(US10047103, 291 | US9688695, 291)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286427(US9518064, Example 43)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175990(US10047103, 23 | US9688695, 23)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175972(US10047103, 5 | US9688695, 5)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176063(US10047103, 96 | US9688695, 96)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600791(CHEMBL5177223)copy SMILES
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176059(US10047103, 92 | US9688695, 92)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176268(US10047103, 301 | US9688695, 301)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600784(CHEMBL5184586)copy SMILES
Affinity DataIC50: 0.630nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286431(US9518064, Example 47)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175989(US10047103, 22 | US9688695, 22)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600790(CHEMBL5171201)copy SMILES
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
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