Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.331nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.603nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranes after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.776nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranes after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]WIN 55212-2 from human CB2 receptor incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
In DepthDetails
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
In DepthDetails
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]-pentazocine from human Sigma 1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1A expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
In DepthDetails
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranes after 150 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University of Modena and Reggio Emilia
Curated by ChEMBL
University of Modena and Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-ditolylguanidine from human Sigma 2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Universit£ degli Studi di Modena e Reggio Emilia
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1B expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair