TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 2.24E+4nMAssay Description:Competitive inhibition of rat intestine sucrase using sucrose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.38E+4nMAssay Description:Competitive inhibition of rat intestine maltase using maltose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 4.75E+4nMAssay Description:Non-competitive inhibition of rat intestine sucrase using sucrose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.45E+4nMAssay Description:Non-competitive inhibition of rat intestine maltase using maltose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.88E+5nMAssay Description:Competitive inhibition of rat intestinal maltase using maltose as substrate assessed as dissociation of enzyme-inhibitor complex at 0.1 to 1 mg/ml by...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 3.80E+5nMAssay Description:Non-competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+5nMAssay Description:Non-competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+5nMAssay Description:Non-competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 5.40E+5nMAssay Description:Non-competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 1.09E+6nMAssay Description:Competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
Affinity DataKi: 1.34E+6nMAssay Description:Non-competitive inhibition of rat intestinal maltase using maltose as substrate assessed as dissociation of enzyme-substrate-inhibitor complex at 0.1...More data for this Ligand-Target Pair
Affinity DataKi: 1.64E+6nMAssay Description:Competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
Affinity DataKi: 1.96E+6nMAssay Description:Competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataKi: 3.07E+6nMAssay Description:Competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat intestinal alpha-glucosidase maltase using maltose as substrate preincubated for 10 mins prior substrate addition measured after 40...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of rat intestinal alpha-glucosidase sucrase using sucrose as substrate preincubated for 10 mins prior substrate addition measured after 40...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.31E+3nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.43E+4nMAssay Description:Inhibition of rat intestinal maltase using maltose as substrate preincubated for 10 mins before substrate addition by glucose oxidase methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.47E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 4.72E+4nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 4.74E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.19E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 6.72E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 8.75E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 9.49E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 1.71E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 3.67E+5nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 4.97E+5nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibition of beta-galactosidaseMore data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 8.05E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University
Curated by ChEMBL
Chulalongkorn University
Curated by ChEMBL
Affinity DataIC50: 9.54E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
Affinity DataIC50: 1.85E+6nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair