Compile Data Set for Download or QSAR
Found 63 with Last Name = 'whiteley' and Initial = 'pe'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15774((2R)-1-({4-[3-(4-fluorophenyl)-1H-pyrrolo[3,2-b]py...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15773((2S)-1-({4-[3-(4-fluorophenyl)-1H-pyrrolo[3,2-b]py...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15776(2-({4-[3-(4-fluorophenyl)-1H-pyrrolo[3,2-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15775(1-({4-[3-(4-fluorophenyl)-1H-pyrrolo[3,2-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15772(4-({4-[3-(4-fluorophenyl)-1H-pyrrolo[3,2-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15756(3-(4-Fluorophenyl)-2-(pyridin-4-yl)-1H-pyrrolo[3,2...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15764(3-(4-Fluorophenyl)-1-methoxy-ethyl-2-pyridin-4-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15765(3-(4-Fluorophenyl)-1-ethyl-2-pyridin-4-yl-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM13531(4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridy...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15759(4,7 Diazaindole 22 | 4-[7-(4-fluorophenyl)-5H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 53nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15763(3-(4-Fluoro-phenyl)-1-methoxy-2-pyridin-4-yl-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 68nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15762(3-(4-Fluorophenyl-2-(pyridin-4yl)furo[3,2-b]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 86nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15766(3-(4-Fluorophenyl)-1-methyl-2-pyridin-4-yl-1H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 98nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15767(1-[3-(4-fluorophenyl)-2-(pyridin-4-yl)-1H-pyrrolo[...)copy SMILEScopy InChI
Affinity DataIC50: 172nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15744(1-(2,4-difluorophenyl)-4-{[3-(pyridin-3-yl)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15768(3-(4-Fluorophenyl)-1-morpholinoethyl-2-pyridin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 185nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15769(3-(4-Fluorophenyl)-1-pyrrolidinoethyl-2-pyridin-4-...)copy SMILEScopy InChI
Affinity DataIC50: 217nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15749(1-[2-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15743(1-(2,4-difluorophenyl)-4-{[3-(pyridin-4-yl)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15745(1-(2,4-difluorophenyl)-4-{[3-(pyridin-3-yloxy)phen...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15750(4-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 590nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15754((2S)-3-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15740(1-(4-fluorophenyl)-4-{[3-(pyridin-3-yl)phenyl]carb...)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15748(1-(4-fluorophenyl)-4-{[3-(2-methanesulfonylethyl)p...)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15746(2-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 850nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15760(4,6 Diazaindole 24 | 4-[7-(4-fluorophenyl)-5H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 895nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15741(1-(4-fluorophenyl)-4-{[4-(pyridin-3-yl)phenyl]carb...)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15718((5-Amino-1-O-tolyl-1H-pyrazol-4-yl)phenylmethanone...)copy SMILEScopy InChI
Affinity DataIC50: 1.08E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15720(4-benzoyl-1-(4-fluorophenyl)-1H-pyrazol-5-amine | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15753((2R)-3-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15747(2-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15725(1-(4-fluorophenyl)-4-({3-[2-(morpholin-4-yl)ethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.27E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15742(1-(4-fluorophenyl)-4-{[3-(pyridin-4-yl)phenyl]carb...)copy SMILEScopy InChI
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15734(1-(4-fluorophenyl)-4-({3-[3-(piperidin-1-yl)prop-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15728(1-(4-fluorophenyl)-4-({3-[2-(4-methylpiperazin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15735(1-(4-fluorophenyl)-4-({3-[3-(morpholin-4-yl)prop-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15737(1-(4-fluorophenyl)-4-({3-[3-(morpholin-4-yl)propyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15758(3-(4-Fluorophenyl)-2-pyridin-4-yl-1H-indole | 3-(4...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15739(1-(4-fluorophenyl)-4-({3-[2-(piperidin-1-yl)ethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15770(3-(4-Fluorophenyl)-1-piperidinoethyl-2-pyridin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.97E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15726(1-(4-fluorophenyl)-4-{[3-(4-methylpiperazin-1-yl)p...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15732(4-({3-[3-(dimethylamino)prop-1-yn-1-yl]phenyl}carb...)copy SMILEScopy InChI
Affinity DataIC50: 2.28E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15714((5-Amino-1-phenyl-1H-pyrazol-4-yl)phenylmethanone ...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15727(4-{[3-(2-aminoethyl)phenyl]carbonyl}-1-(4-fluoroph...)copy SMILEScopy InChI
Affinity DataIC50: 2.44E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15733(1-(4-fluorophenyl)-4-({3-[3-(4-methylpiperazin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15722(4-benzoyl-1-(2-fluorophenyl)-1H-pyrazol-5-amine | ...)copy SMILEScopy InChI
Affinity DataIC50: 2.86E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15757(3-(4-Fluorophenyl)-2-pyridin-4-yl)-1H-pyrrolo[3,2-...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15736(1-(4-fluorophenyl)-4-({4-[3-(morpholin-4-yl)prop-1...)copy SMILEScopy InChI
Affinity DataIC50: 3.13E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15761(7-(4-Fluoro-phenyl)-6-pyridin-4-yl-7H-pyrrolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMpH: 7.4 T: 2°CAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6QHTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Roche Palo Alto LLC

LigandPNGBDBM15751(1-(3-{[5-amino-1-(4-fluorophenyl)-1H-pyrazol-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant active p38alpha MAP kinase was tested by measuring the incorporation of 33P from gamma-[33P] ATP into myelin basic pr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23776ZNPubMed
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