Compile Data Set for Download or QSAR
Found 101 with Last Name = 'ciaccio' and Initial = 'pj'
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032651(1-((1S,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-y...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344250(CHEMBL1779003 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344232(1-cyclopropyl-N-((6-(4-fluoro-2-methoxyphenyl)pyra...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344251(CHEMBL1779004 | N-((4'-fluoro-2'-methoxybiphenyl-3...)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344233(CHEMBL1778866 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344234(CHEMBL1778867 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  54nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344252(CHEMBL1779005 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344259(CHEMBL1779012 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344254(CHEMBL1779007 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344260(CHEMBL1779013 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344241(CHEMBL1778994 | N-((6-(2,3-difluorophenyl)pyrazin-...)copy SMILEScopy InChI
Affinity DataKi:  186nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344235(CHEMBL1778868 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  214nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344236(CHEMBL1778869 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  217nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344237(CHEMBL1778870 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  255nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344255(CHEMBL1779008 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  266nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344262(CHEMBL1779015 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  268nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344264(CHEMBL1779016 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344242(1-cyclopropyl-N-((6-(2,3-difluorophenyl)pyrazin-2-...)copy SMILEScopy InChI
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344265(3-((5-(4-fluoro-2-methoxyphenyl)pyridin-3-yl)methy...)copy SMILEScopy InChI
Affinity DataKi:  420nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344238(CHEMBL1778991 | N-((6-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  429nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344256(3-(4-fluoro-2-methoxyphenyl)-5-(pyrrolidin-2-yl)py...)copy SMILEScopy InChI
Affinity DataKi:  440nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344261(CHEMBL1779014 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  450nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344257(CHEMBL1779010 | N-benzyl-5-(4-fluoro-2-methoxyphen...)copy SMILEScopy InChI
Affinity DataKi:  457nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344266(CHEMBL1779018 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  468nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344267(CHEMBL1779019 | N-((5-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  595nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344244(1-cyclopropyl-N-((6-(2-fluoro-3-methoxyphenyl)pyra...)copy SMILEScopy InChI
Affinity DataKi:  602nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344239((S)-1-(6-(4-fluoro-2-methoxyphenyl)pyrazin-2-yl)-N...)copy SMILEScopy InChI
Affinity DataKi:  610nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344258(5-(4-fluoro-2-methoxyphenyl)-N-(tetrahydro-2H-pyra...)copy SMILEScopy InChI
Affinity DataKi:  705nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344268(CHEMBL1779020 | ethyl 2-((5-(4-fluoro-2-methoxyphe...)copy SMILEScopy InChI
Affinity DataKi:  778nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344246(3-(6-((cyclopentylamino)methyl)pyrazin-2-yl)benzon...)copy SMILEScopy InChI
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344247(4-(6-((cyclopentylamino)methyl)pyrazin-2-yl)benzon...)copy SMILEScopy InChI
Affinity DataKi:  1.57E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344248(CHEMBL1779001 | N-((6-(2,4-dimethoxyphenyl)pyrazin...)copy SMILEScopy InChI
Affinity DataKi:  1.69E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344243(CHEMBL1778996 | N-((6-(2,3-difluorophenyl)pyrazin-...)copy SMILEScopy InChI
Affinity DataKi:  2.98E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344240(1-(6-(4-fluoro-2-methoxyphenyl)pyrazin-2-yl)-N-(py...)copy SMILEScopy InChI
Affinity DataKi:  3.57E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344245(CHEMBL1778998 | N-((6-(2-fluoro-3-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  5.70E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344253(CHEMBL1779006 | N-((2-(4-fluoro-2-methoxyphenyl)py...)copy SMILEScopy InChI
Affinity DataKi:  8.90E+3nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
AstraZeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50344249(CHEMBL1779002 | N-(3-(6-((cyclopentylamino)methyl)...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP101606 from NR2B in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29887BKPubMed
LigandPNGBDBM50584324(CHEMBL5088471)copy SMILES
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584332(CHEMBL5076397)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584325(CHEMBL5085777)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584321(CHEMBL5090739)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584318(CHEMBL5082563)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584331(CHEMBL5079796)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584330(CHEMBL5070497)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584328(CHEMBL5078277 | US20230303540, Example Ex-1.48)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584316(CHEMBL5070231)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584317(CHEMBL5082260)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584322(CHEMBL5089102)copy SMILES
Affinity DataIC50: 0.650nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584326(CHEMBL5094138)copy SMILES
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584320(CHEMBL5073571)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
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