Compile Data Set for Download or QSAR
Found 334 with Last Name = 'depue' and Initial = 'pl'
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of ET-1 binding to Endothelin A receptor in cultured rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1XGJPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ET-1 binding to Endothelin B receptor in cultured rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1XGJPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032181(2-{1-[1-(2-carboxy-1-{1-[10,11-dihydro-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032175((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032181(2-{1-[1-(2-carboxy-1-{1-[10,11-dihydro-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032175((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032216((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032193((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032175((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of ET-1 binding to Endothelin A receptor in cultured rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1XGJPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032181(2-{1-[1-(2-carboxy-1-{1-[10,11-dihydro-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032202((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032207((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in CHO cells expressing rat ET- B receptorsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032166((S)-3-[(S)-2-((S)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032178((S)-N-((1S,2S)-1-{(1S,2S)-1-[(S)-1-Carboxy-2-(1H-i...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in CHO cells expressing rat ET- B receptorsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032191((S)-4-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032171((S)-4-((S)-2-Acetylamino-3,3-diphenyl-propionylami...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B/1 receptor(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032207((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50281565((S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908MP
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032193((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032173((S)-3-[(S)-2-((S)-2-Benzoylamino-3,3-diphenyl-prop...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032180((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032202((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045240((S)-2-[(S)-2-((2S,5S)-2-{(S)-2-[(S)-2-((R)-2-Acety...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908MP
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045240((S)-2-[(S)-2-((2S,5S)-2-{(S)-2-[(S)-2-((R)-2-Acety...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032198((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032198((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Binding affinity measured in CHO cells stably transfected with the human endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B/1 receptor(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045244((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-ET-1 from Endothelin B receptor of rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908MP
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032207((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032171((S)-4-((S)-2-Acetylamino-3,3-diphenyl-propionylami...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032208((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Binding affinity against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50284007(CHEMBL412460 | Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Se...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4QW6
TargetEndothelin receptor type B(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Binding affinity against endothelin B receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045244((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032191((S)-4-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045244((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032216((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032172((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032202((S)-2-[(2S,3S)-2-((2S,3S)-2-{(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Effective concentration against Endothelin B receptor from rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69K6KPubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032201((S)-2-((2S,3S)-2-{(2S,3S)-2-[(S)-2-[(S)-2-((S)-2-A...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032186((S)-3-[(S)-2-((S)-2-Acetylamino-3,3-diphenyl-propi...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50032171((S)-4-((S)-2-Acetylamino-3,3-diphenyl-propionylami...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KD1WZQPubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50001220(3-{2-[2-Acetylamino-3-(1H-indol-3-yl)-propionylami...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of ET-1 binding to Endothelin A receptor in cultured rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1XGJPubMed
Displayed 1 to 50 (of 334 total ) | Next | Last >>
Jump to: