Compile Data Set for Download or QSAR
Found 207 with Last Name = 'beardsley' and Initial = 'pm'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001090(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001088((DPDPE)13-[2-Amino-3-(4-hydroxy-phenyl)-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001090(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Dissociation rate constant of compound for mutant T46S Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86208(cis-CPCA, -)copy SMILEScopy InChI
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetNorepinephrine transporter(RAT)
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86206(CAS_8268 | CPCA, + | NSC_8268)copy SMILEScopy InChI
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001091(10-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Dissociation rate constant of compound for mutant T46A Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001091(10-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetNorepinephrine transporter(RAT)
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86208(cis-CPCA, -)copy SMILEScopy InChI
Affinity DataKi:  98nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetNorepinephrine transporter(RAT)
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86207(CAS_50-36-2 | COCAINE | NSC_446220)copy SMILEScopy InChI
Affinity DataKi:  119nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001091(10-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001091(10-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86207(CAS_50-36-2 | COCAINE | NSC_446220)copy SMILEScopy InChI
Affinity DataKi:  177nMMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86207(CAS_50-36-2 | COCAINE | NSC_446220)copy SMILEScopy InChI
Affinity DataKi:  275nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86206(CAS_8268 | CPCA, + | NSC_8268)copy SMILEScopy InChI
Affinity DataKi:  276nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle and Company

Curated by ChEMBL
LigandPNGBDBM50001088((DPDPE)13-[2-Amino-3-(4-hydroxy-phenyl)-propionyla...)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7QF6PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM86206(CAS_8268 | CPCA, + | NSC_8268)copy SMILEScopy InChI
Affinity DataKi:  5.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R20ZZ8PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50125902((1S,4R)-4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benz...)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)copy SMILEScopy InChI
Affinity DataIC50: 0.960nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50055876(4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benzyl)-pipe...)copy SMILEScopy InChI
Affinity DataIC50: 2.48nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108818(4-(2-Benzhydryloxy-ethyl)-1-(4-vinyl-benzyl)-piper...)copy SMILEScopy InChI
Affinity DataIC50: 2.96nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50098393(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)copy SMILEScopy InChI
Affinity DataIC50: 3.67nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50125902((1S,4R)-4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benz...)copy SMILEScopy InChI
Affinity DataIC50: 4.05nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108817(4-(2-Benzhydryloxy-ethyl)-1-(4-ethynyl-benzyl)-pip...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50098396(Benzhydryl-[2-(1-benzyl-piperidin-4-yl)-ethyl]-ami...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50098396(Benzhydryl-[2-(1-benzyl-piperidin-4-yl)-ethyl]-ami...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 6.63nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50098395(Benzhydryl-{2-[1-(3,4-difluoro-benzyl)-piperidin-4...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108823(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)copy SMILEScopy InChI
Affinity DataIC50: 8.23nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50066414(Benzhydryl-{2-[1-(4-fluoro-benzyl)-piperidin-4-yl]...)copy SMILEScopy InChI
Affinity DataIC50: 9.37nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50125905((3R,4S)-4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benz...)copy SMILEScopy InChI
Affinity DataIC50: 10.1nMAssay Description:Inhibition of uptake from dopamine transporter in rat striatum using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50098397(4-(2-Benzhydryloxy-ethyl)-1-(3,4-difluoro-benzyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 10.1nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 10.6nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40P0PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 10.6nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 10.6nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 10.6nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50154243(4-[(6-Benzhydryl-piperidin-3-ylamino)-methyl]-benz...)copy SMILEScopy InChI
Affinity DataIC50: 11.2nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ40P0PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50125905((3R,4S)-4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benz...)copy SMILEScopy InChI
Affinity DataIC50: 11.2nMAssay Description:Binding affinity towards dopamine transporter in rat striatum using [3H]WIN-35 428 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37XTPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108820(4-(2-Benzhydryloxy-ethyl)-1-(4-isopropenyl-benzyl)...)copy SMILEScopy InChI
Affinity DataIC50: 11.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50108821(3-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)copy SMILEScopy InChI
Affinity DataIC50: 14.3nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FJ2HHVPubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University

Curated by PDSP Ki Database
LigandPNGBDBM50055876(4-(2-Benzhydryloxy-ethyl)-1-(4-fluoro-benzyl)-pipe...)copy SMILEScopy InChI
Affinity DataIC50: 17.2nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20002SRPubMed
Displayed 1 to 50 (of 207 total ) | Next | Last >>
Jump to: