Compile Data Set for Download or QSAR
Found 70 with Last Name = 'sunderland' and Initial = 'pt'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341860(8-chloro-2-(4-(4-(4-fluorophenyl)-5,6-dihydropyrid...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341859(2-(4-chlorophenyl)quinoxaline-5-carboxamide | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341859(2-(4-chlorophenyl)quinoxaline-5-carboxamide | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of calf thymus PARP-1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438600(CHEMBL2414048)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of PARP-1 (unknown origin) in broken nuclear preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438608(CHEMBL2414049)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438605(CHEMBL2414042)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)copy SMILEScopy InChI
Affinity DataIC50: 490nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341860(8-chloro-2-(4-(4-(4-fluorophenyl)-5,6-dihydropyrid...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341856(5-(Carboxymethylamino)isoquinolin-1-one | CHEMBL17...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341857(5-Amino-2-(2-carboxyethyl)isoquinolin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438601(CHEMBL2414046)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438599(CHEMBL2414051)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438603(CHEMBL2414044)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438602(CHEMBL2414045)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 940nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of mouse PARP-2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438604(CHEMBL2414043)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438606(CHEMBL2414052)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341867(5-(4-Iodobenzamido)isoquinolin-1-one | CHEMBL17670...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341861(5-Benzamidoisoquinolin-1-one | CHEMBL1767054)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM39220((1-oxidanylidene-2H-isoquinolin-5-yl) benzoate | (...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341857(5-Amino-2-(2-carboxyethyl)isoquinolin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341856(5-(Carboxymethylamino)isoquinolin-1-one | CHEMBL17...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341863(5-(4-Nitrobenzamido)isoquinolin-1-one | CHEMBL1767...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341877(3-(1-Oxoisoquinolin-5-yl)propanoic acid | CHEMBL17...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341863(5-(4-Nitrobenzamido)isoquinolin-1-one | CHEMBL1767...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341869(5-(2-Iodobenzamido)isoquinolin-1-one | CHEMBL17670...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341864(5-(4-Trifluoromethylbenzamido)isoquinolin-1-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341865(5-(4-Fluorobenzamido)isoquinolin-1-one | CHEMBL176...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341866(5-(4-Chlorobenzamido)isoquinolin-1-one | CHEMBL176...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM39220((1-oxidanylidene-2H-isoquinolin-5-yl) benzoate | (...)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341869(5-(2-Iodobenzamido)isoquinolin-1-one | CHEMBL17670...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of full length human PARP-1 after 10 mins by FlashPlate scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341876(CHEMBL1767063 | E-3-(1-Oxoisoquinolin-5-yl)propeno...)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438607(CHEMBL2414050)copy SMILEScopy InChI
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341868(5-(2-Methylbenzamido)isoquinolin-1-one | CHEMBL176...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50438609(CHEMBL2414047)copy SMILEScopy InChI
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of human PARP-1 assessed as synthesis of [3H]-ADP-ribose polymers from [3H]-NAD+ by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341874(5-Benzamido-3-methylisoquinolin-1-one | CHEMBL1767...)copy SMILEScopy InChI
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
TargetPoly [ADP-ribose] polymerase 2(Mus musculus (Mouse))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50341862(5-(4-Methylbenzamido)isoquinolin-1-one | CHEMBL176...)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of recombinant full length mouse PARP-2 after 10 mins using [3H]NAD+ by solution-phase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B31NCPubMed
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