Affinity DataKi: 0.350nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.85nMAssay Description:Binding affinity to monkey bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.18nMAssay Description:Binding affinity to rat bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to rabbit bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24.5nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 59.1nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71.5nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 83.5nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 88.5nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Binding affinity to dog bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 479nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 516nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 579nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+3nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.93nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.47nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.65nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.65nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of p110alpha/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
Affinity DataIC50: 43.6nMAssay Description:Binding affinity to human bradikinin B1 receptor by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of mTORC1 (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of p110alpha/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of mTORC1 (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of p110beta/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 148nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Xi'an Jiaotong University
Curated by ChEMBL
Xi'an Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 478nMAssay Description:Inhibition of p110beta/p85alpha (unknown origin) incubated for 40 mins by luciferase based ATP depletion assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
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