Compile Data Set for Download or QSAR
Found 32 with Last Name = 'ang' and Initial = 'qa'
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)copy SMILEScopy InChI
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)copy SMILEScopy InChI
Affinity DataKi:  4.58E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetReplicase polyprotein 1ab(2019-nCoV)TBA
LigandPNGBDBM50599200(CHEMBL5182995 | US11753373, Compound D-1-c)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(2019-nCoV)TBA
LigandPNGBDBM50599197(CHEMBL5173582 | US11753373, Compound D-1-f)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599200(CHEMBL5182995 | US11753373, Compound D-1-c)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599197(CHEMBL5173582 | US11753373, Compound D-1-f)copy SMILES
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(2019-nCoV)TBA
LigandPNGBDBM496902(CVD-0018409 | PF-07321332 | US11351149, Example 13...)copy SMILEScopy InChI
Affinity DataIC50: 31nMMore data for this Ligand-Target Pair
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599203(CHEMBL5183165)copy SMILES
Affinity DataIC50: 70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM496902(CVD-0018409 | PF-07321332 | US11351149, Example 13...)copy SMILEScopy InChI
Affinity DataIC50: 145nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM535146(WO2022013684, Example 13)copy SMILES
Affinity DataIC50: 239nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599202(CHEMBL5173858)copy SMILES
Affinity DataIC50: 290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599204(CHEMBL5174632)copy SMILES
Affinity DataIC50: 467nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026058(CHEMBL3335259)copy SMILEScopy InChI
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM10620((S)-3-(1-(dimethylamino)ethyl)phenyl ethyl(methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026061(CHEMBL3335261)copy SMILEScopy InChI
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026062(CHEMBL3335256)copy SMILEScopy InChI
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026064(CHEMBL3335258)copy SMILEScopy InChI
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026065(CHEMBL3335255)copy SMILEScopy InChI
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026063(CHEMBL3335257)copy SMILEScopy InChI
Affinity DataIC50: 5.48E+4nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599201(CHEMBL5208243)copy SMILES
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599199(CHEMBL5178853)copy SMILES
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599198(CHEMBL5207993)copy SMILES
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetReplicase polyprotein 1ab(HCoV-229E)TBA
LigandPNGBDBM50599196(CHEMBL5199404)copy SMILES
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50S0KPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Hunan University

Curated by ChEMBL
LigandPNGBDBM50026060(CHEMBL3335260)copy SMILEScopy InChI
Affinity DataIC50: 2.65E+5nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate preincubated for 25 mins by Ellman's/UV-vis spectroscopy analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XKVPubMed