Compile Data Set for Download or QSAR
Found 229 with Last Name = 'guo' and Initial = 'ql'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of cSrc (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMedDrugBank
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMedDrugBank
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMedDrugBank
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271947(6-Methoxy-7-[2-(4-methylpiperazin-1-yl)-ethoxy]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 9.23nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351284(CHEMBL1818768)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271896(6-Methyl-7-[3-(piperidin-1-yl)-propoxy]-4-(6-methy...)copy SMILEScopy InChI
Affinity DataIC50: 15.4nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271896(6-Methyl-7-[3-(piperidin-1-yl)-propoxy]-4-(6-methy...)copy SMILEScopy InChI
Affinity DataIC50: 15.4nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetCholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human serum BuChE using butylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for 2 min...More data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351271(CHEMBL1818755)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275877(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methoxy-7-(...)copy SMILEScopy InChI
Affinity DataIC50: 20.7nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351274(CHEMBL1818758)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351290(CHEMBL1818774)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for...More data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351283(CHEMBL1818767)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275756(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(2...)copy SMILEScopy InChI
Affinity DataIC50: 34.8nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275812(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)copy SMILEScopy InChI
Affinity DataIC50: 36.6nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275813(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(diethyl...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351272(CHEMBL1818756)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351289(CHEMBL1818773)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275757(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)copy SMILEScopy InChI
Affinity DataIC50: 50.6nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351259(CHEMBL1818674)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50198311((R)-N-(1-(3-benzyl-7-chloro-4-oxo-3,4-dihydroquina...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275811(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)copy SMILEScopy InChI
Affinity DataIC50: 53.4nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351288(CHEMBL1818772)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271839(6-Methyl-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 75.9nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275758(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)copy SMILEScopy InChI
Affinity DataIC50: 81.1nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351282(CHEMBL1818766)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271897(6-Methyl-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 111nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275759(4-(2-aminobenzo[d]thiazol-6-ylamino)-6-methyl-7-(3...)copy SMILEScopy InChI
Affinity DataIC50: 129nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271948(6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4...)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275875(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-7-(3-(di...)copy SMILEScopy InChI
Affinity DataIC50: 143nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351270(CHEMBL1818754)copy SMILEScopy InChI
Affinity DataIC50: 146nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351281(CHEMBL1818765)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275876(4-(2-amino-1H-benzo[d]imidazol-6-ylamino)-6-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 159nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351277(CHEMBL1818761)copy SMILEScopy InChI
Affinity DataIC50: 162nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351279(CHEMBL1818763)copy SMILEScopy InChI
Affinity DataIC50: 169nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351280(CHEMBL1818764)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271840(6-Methyl-7-(3-morpholinopropoxy)-4-(benzothiazol-2...)copy SMILEScopy InChI
Affinity DataIC50: 172nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271900(6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4...)copy SMILEScopy InChI
Affinity DataIC50: 178nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271899(6-Methoxy-7-[3-(4-methylpiperazin-1-yl)-propoxy]-4...)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271841(6-Methyl-7-[3-(piperidin-1-yl)-propoxy]-4-(benzoth...)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351263(CHEMBL1818747)copy SMILEScopy InChI
Affinity DataIC50: 232nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50275814(4-(2-aminobenzo[d]thiazol-6-ylamino)-7-(3-(3,5-dim...)copy SMILEScopy InChI
Affinity DataIC50: 267nMAssay Description:Inhibition of cSrc (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K0743JPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM93333(Met-33)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55R0JPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for...More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50264634(CHEMBL4067639)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human serum BuChE using butylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55R0JPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351260(CHEMBL1818675)copy SMILEScopy InChI
Affinity DataIC50: 334nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50351262(CHEMBL1818677)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of human ATPase activity KSP expressed in Escherichia coli after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B858HDPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50271945(6-Methoxy-7-[2-(piperidin-1-yl)-ethoxyl]-4-(benzot...)copy SMILEScopy InChI
Affinity DataIC50: 371nMAssay Description:Inhibition of human recombinant cSrc by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60PZ6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50264600(CHEMBL4066392)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine chloride as substrate pretreated for 15 mins followed by substrate addition measured for...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55R0JPubMed
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