Compile Data Set for Download or QSAR
Found 382 with Last Name = 'chambers' and Initial = 'r'
TargetPlasma kallikrein(Homo sapiens (Human))TBA
LigandPNGBDBM50579244(Avoralstat | BCX-4161)copy SMILES
Affinity DataKi:  0.260nMAssay Description:Inhibition of purified human plasma kallikrein assessed as inhibition constant using H-D-Pro-Phe-Arg-pNA.2HCl as substrate measured after 3 mins by m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C7288PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50081533(CHEMBL96224 | CP-199331 | N-{3-[(3R,4R)-6-(5,6-Dif...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MP52G3PubMed
TargetPlasma kallikrein(Homo sapiens (Human))TBA
LigandPNGBDBM416926((+)-1-(3-(aminomethyl)phenyl)-N-(5-((3-cyanophenyl...)copy SMILEScopy InChI
Affinity DataKi:  0.440nMAssay Description:Inhibition of purified human plasma kallikrein assessed as inhibition constant using H-D-Pro-Phe-Arg-pNA.2HCl as substrate measured after 3 mins by m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C7288PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50081532(CHEMBL96206 | CP-199330 | N-{3-[(3R,4R)-6-(7-Chlor...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MP52G3PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070919(C,C,C-Trifluoro-N-{3-[(2R,3S,4R)-6-(5-fluoro-benzo...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50023198(8-[4-(4-phenylbutyloxy)benzoyl]amino-2-(tetrazol-5...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50023198(8-[4-(4-phenylbutyloxy)benzoyl]amino-2-(tetrazol-5...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50023198(8-[4-(4-phenylbutyloxy)benzoyl]amino-2-(tetrazol-5...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Compound was evaluated in vitro for the binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50073277(CHEMBL332680 | N-{3-[(3S,4R)-6-(5,6-Difluoro-benzo...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070919(C,C,C-Trifluoro-N-{3-[(2R,3S,4R)-6-(5-fluoro-benzo...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Compound was evaluated in vitro for the binding of cysLT1 receptor to guinea pig lung membranes.More data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070919(C,C,C-Trifluoro-N-{3-[(2R,3S,4R)-6-(5-fluoro-benzo...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50215874(CHEMBL52102)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50073279(CHEMBL119214 | N-{3-[(3S,4R)-6-(7-Chloro-quinolin-...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50073276(CHEMBL120200 | N-{4-Chloro-3-[(3S,4R)-6-(5,6-diflu...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50073275(CHEMBL331884 | N-(3-{(3S,4R)-6-[(E)-2-(7-Chloro-qu...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50073278(CHEMBL331747 | N-{3-[(3S,4R)-6-(5,6-Difluoro-benzo...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070921(3-[(3R,4R)-6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2833R5MPubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070921(3-[(3R,4R)-6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50215871(CHEMBL415954)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284689(7-Chloro-2-((E)-2-{3-[4-(2-methyl-imidazo[4,5-c]py...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LTD4 from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284689(7-Chloro-2-((E)-2-{3-[4-(2-methyl-imidazo[4,5-c]py...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50215875(CHEMBL299779)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284691(2-(2-{3-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-p...)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284690(1-(4-{3-[(E)-2-(5-Fluoro-benzothiazol-2-yl)-vinyl]...)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284690(1-(4-{3-[(E)-2-(5-Fluoro-benzothiazol-2-yl)-vinyl]...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284691(2-(2-{3-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-p...)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50215872(CHEMBL50399)copy SMILEScopy InChI
Affinity DataKi:  92nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50215873(CHEMBL297906)copy SMILEScopy InChI
Affinity DataKi:  434nMAssay Description:Ability to antagonize LTD4 receptors isolated from guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N3004BPubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284680((3S,4S)-3-Pyridin-3-ylmethyl-6-(quinolin-2-ylmetho...)copy SMILEScopy InChI
Affinity DataKi:  650nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5NSM
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284682(2-Benzyl-7-(quinolin-2-ylmethoxy)-1,2,3,4-tetrahyd...)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5NSM
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50284681(2-Butyl-7-(quinolin-2-ylmethoxy)-1,2,3,4-tetrahydr...)copy SMILEScopy InChI
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5NSM
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50012434((REV-5,901)1-[3-(Quinolin-2-ylmethoxy)-phenyl]-hex...)copy SMILEScopy InChI
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5NSM
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50070921(3-[(3R,4R)-6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4...)copy SMILEScopy InChI
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5NSM
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-leukotriene D4 (LTD4) from receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-ligand from platelet activating factor (PAF) receptor in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M045D5
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282990(CHEMBL59973 | Morpholine-4-carboxylic acid ((S)-1-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for the inhibition of human plasma renin(Hu Renin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8CQ7
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50104526(3-[2-((S)-3-Methyl-1-{2-[4-(3-o-tolyl-ureido)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human recombinant sVCAM-1 binding to alpha4-beta1 integrin (VLA-4) in ELISAMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41SQZPubMed
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282993((2S,4R)-4-Cyclohexyl-2-hydroxy-3-((R)-3-methylsulf...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Compound was tested for the inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8CQ7
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50071637(CHEMBL79366 | {1-Dimethylcarbamoyl-3-[2-methoxy-4-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63M30PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50071633(CHEMBL83166 | [3-[2-Methoxy-4-(toluene-2-sulfonyla...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63M30PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50071631(CHEMBL79952 | [3-[2-Methoxy-4-(toluene-2-sulfonyla...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63M30PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50071632(CHEMBL310446 | {1-Diethylcarbamoyl-3-[2-methoxy-4-...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63M30PubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50071636(CHEMBL79479 | {1-(2-Dimethylamino-ethylcarbamoyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against leukotriene D4 receptor in [3H]-LTD4 binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63M30PubMed
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282993((2S,4R)-4-Cyclohexyl-2-hydroxy-3-((R)-3-methylsulf...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Compound was tested for the inhibition of monkey plasma reninMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8CQ7
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282993((2S,4R)-4-Cyclohexyl-2-hydroxy-3-((R)-3-methylsulf...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Compound was tested for the inhibition of guinea pig plasma reninMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8CQ7
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